Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 6404
TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126820(US8785477, 26)
Affinity DataIC50: 2.61nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126816(US8785477, 8)
Affinity DataIC50: 11.2nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126818(US8785477, 17)
Affinity DataIC50: 11.5nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
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Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126815(US8785477, 3)
Affinity DataIC50: 17.7nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
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Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126814(US8785477, 1)
Affinity DataIC50: 22.8nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
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Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126819(US8785477, 20)
Affinity DataIC50: 23.2nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126817(US8785477, 12)
Affinity DataIC50: 25.9nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
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TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126822(US8785477, Sitagliptin)
Affinity DataIC50: 26.0nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
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PDB3D3D Structure (crystal)
TargetDipeptidyl peptidase 4(Rat)
Shanghai Sun-Sail Pharmaceutical Science & Technology

US Patent
LigandPNGBDBM126821(US8785477, Vildagliptin)
Affinity DataIC50: 80.1nMAssay Description:Thoroughly mixed test compounds, enzyme and reaction buffer, preincubated the mixture for 15 minutes at 37° C. and then primed reaction by adding sub...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/16/2014
Entry Details
Go to US Patent