Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 6389
TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125988BDBM125988(US8772297, Y244)
Affinity DataIC50: 600nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125985BDBM125985(US8772297, Y241)
Affinity DataIC50: 700nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125986BDBM125986(US8772297, Y260)
Affinity DataIC50: 1.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125979BDBM125979(US8772297, Y177)
Affinity DataIC50: 2.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125980BDBM125980(US8772297, Y224)
Affinity DataIC50: 2.40E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125989BDBM125989(US8772297, Y250)
Affinity DataIC50: 2.50E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125981BDBM125981(US8772297, Y186)
Affinity DataIC50: 3.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125991BDBM125991(US8772297, Y296)
Affinity DataIC50: 4.60E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125990BDBM125990(US8772297, Y284)
Affinity DataIC50: 6.70E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125987BDBM125987(US8772297, Y366)
Affinity DataIC50: 7.30E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125976BDBM125976(US8772297, Y145)
Affinity DataIC50: 8.00E+3nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125978BDBM125978(US8772297, Y155)
Affinity DataIC50: 1.40E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125982BDBM125982(US8772297, Y178)
Affinity DataIC50: 1.50E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125984BDBM125984(US8772297, Y196)
Affinity DataIC50: 1.60E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125973BDBM125973(US8772297, Y141)
Affinity DataIC50: 1.70E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125977BDBM125977(US8772297, Y147)
Affinity DataIC50: 1.80E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125974BDBM125974(US8772297, Y142)
Affinity DataIC50: 2.20E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125983BDBM125983(US8772297, Y185)
Affinity DataIC50: 2.40E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125972BDBM125972(US8772297, Y098)
Affinity DataIC50: 2.70E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent

TargetTGF-beta receptor type-1(Human)
Kyoto University

US Patent
LigandChemical structure of BindingDB Monomer ID 125975BDBM125975(US8772297, Y140)
Affinity DataIC50: 3.00E+4nMAssay Description:The biological activity of a compound was determined by measuring the activation of Smad3/Smad4 complex which is a transcription factor showing activ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2014
Entry Details
US Patent