Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 6330
TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123468(US8748626, 1)
Affinity DataIC50: 0.840nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
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TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123472(US8748626, 5)
Affinity DataIC50: 2.54nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123470(US8748626, 3)
Affinity DataIC50: 2.60nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123471(US8748626, 4)
Affinity DataIC50: 7.18nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123469(US8748626, 2)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123475(US8748626, 8)
Affinity DataIC50: 216nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123474(US8748626, 7)
Affinity DataIC50: 631nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent

TargetKinesin-like protein KIF11(Human)
Novartis

US Patent
LigandPNGBDBM123473(US8748626, 6)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:This example provides a representative in vitro assay for determining KSP activity in vitro. Purified microtubules obtained from bovine brain were pu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/5/2014
Entry Details
Go to US Patent