Compile Data Set for Download or QSAR
Report error Found 248 Enz. Inhib. hit(s) with all data for entry = 6314
TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122478(US8729061, 8)
Affinity DataIC50: 0.296nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122498(US8729061, 28)
Affinity DataIC50: 0.328nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122508(US8729061, 38)
Affinity DataIC50: 0.340nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122479(US8729061, 9)
Affinity DataIC50: 0.367nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122495(US8729061, 25)
Affinity DataIC50: 0.403nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122486(US8729061, 16)
Affinity DataIC50: 0.442nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122528(US8729061, 58)
Affinity DataIC50: 0.478nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122513(US8729061, 43)
Affinity DataIC50: 0.508nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122485(US8729061, 15)
Affinity DataIC50: 0.520nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122518(US8729061, 48)
Affinity DataIC50: 0.527nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122494(US8729061, 24)
Affinity DataIC50: 0.550nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122509(US8729061, 39)
Affinity DataIC50: 0.558nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122490(US8729061, 20)
Affinity DataIC50: 0.560nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122511(US8729061, 41)
Affinity DataIC50: 0.568nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122489(US8729061, 19)
Affinity DataIC50: 0.593nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122488(US8729061, 18)
Affinity DataIC50: 0.600nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122524(US8729061, 54)
Affinity DataIC50: 0.630nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122512(US8729061, 42)
Affinity DataIC50: 0.634nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122487(US8729061, 17)
Affinity DataIC50: 0.652nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122484(US8729061, 14)
Affinity DataIC50: 0.668nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122491(US8729061, 21)
Affinity DataIC50: 0.668nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122523(US8729061, 53)
Affinity DataIC50: 0.676nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122483(US8729061, 13)
Affinity DataIC50: 0.704nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122502(US8729061, 32)
Affinity DataIC50: 0.734nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122482(US8729061, 12)
Affinity DataIC50: 0.737nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122506(US8729061, 36)
Affinity DataIC50: 0.776nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122514(US8729061, 44)
Affinity DataIC50: 0.779nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122504(US8729061, 34)
Affinity DataIC50: 0.787nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122501(US8729061, 31)
Affinity DataIC50: 0.827nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122471(US8729061, 1)
Affinity DataIC50: 0.829nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122525(US8729061, 55)
Affinity DataIC50: 0.876nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetProcathepsin L(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122528(US8729061, 58)
Affinity DataIC50: 0.900nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122519(US8729061, 49)
Affinity DataIC50: 0.901nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122476(US8729061, 6)
Affinity DataIC50: 0.976nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122492(US8729061, 22)
Affinity DataIC50: 0.983nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122473(US8729061, 3)
Affinity DataIC50: 1.00nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122507(US8729061, 37)
Affinity DataIC50: 1.02nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122510(US8729061, 40)
Affinity DataIC50: 1.06nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122503(US8729061, 33)
Affinity DataIC50: 1.11nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122472(US8729061, 2)
Affinity DataIC50: 1.12nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122505(US8729061, 35)
Affinity DataIC50: 1.21nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122499(US8729061, 29)
Affinity DataIC50: 1.26nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122481(US8729061, 11)
Affinity DataIC50: 1.38nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122500(US8729061, 30)
Affinity DataIC50: 1.42nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetProcathepsin L(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122523(US8729061, 53)
Affinity DataIC50: 1.70nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122475(US8729061, 5)
Affinity DataIC50: 1.83nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122522(US8729061, 52)
Affinity DataIC50: 1.96nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetProcathepsin L(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122519(US8729061, 49)
Affinity DataIC50: 2nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122532(US8729061, 62)
Affinity DataIC50: 2.35nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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TargetCathepsin S(Human)
Hoffmann-La Roche

US Patent
LigandPNGBDBM122526(US8729061, 56)
Affinity DataIC50: 2.57nMpH: 6.5Assay Description:Enzyme activity is measured by observing the increase in fluorescence intensity caused by cleavage of a peptide substrate containing a fluorophore wh...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2014
Entry Details
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