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Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 6274
TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50393560(CHEMBL2158300 | US8697716, 48)
Affinity DataIC50: 5nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120083(US8697716, 52)
Affinity DataIC50: 8nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120084(US8697716, 55)
Affinity DataIC50: 12nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50393539(CHEMBL2158225 | US8697716, 26)
Affinity DataIC50: 26nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120085(US8697716, 56)
Affinity DataIC50: 39nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120080(US8697716, 38)
Affinity DataIC50: 39nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120075(US8697716, 8)
Affinity DataIC50: 42nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120077(US8697716, 21)
Affinity DataIC50: 50nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50393544(CHEMBL2158230 | US8697716, 34)
Affinity DataIC50: 52nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120076(CHEMBL256712 | US8697716, 16)
Affinity DataIC50: 57nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50377058(CHEMBL2158221 | CHEMBL257154 | US8697716, 14)
Affinity DataIC50: 71nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120079(CHEMBL257153 | US8697716, 35)
Affinity DataIC50: 73nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120078(US8697716, 27)
Affinity DataIC50: 80nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120082(US8697716, 47)
Affinity DataIC50: 100nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50377066(CHEMBL265432 | US8697716, 11)
Affinity DataIC50: 150nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM120081(US8697716, 40)
Affinity DataIC50: 160nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMast/stem cell growth factor receptor Kit(Human)
Janssen Pharmaceutica

US Patent
LigandPNGBDBM50377067(CHEMBL427775 | US8697716, 12)
Affinity DataIC50: 250nMAssay Description:The compounds of the present invention are also specific inhibitors of c-Kit. Selection of preferred compounds of Formula I for use as c-Kit inhibito...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
Go to US Patent