Compile Data Set for Download or QSAR
Report error Found 866 Enz. Inhib. hit(s) with all data for entry = 6278
TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120258(US8691753, 95 bis)
Affinity DataKi:  0.300nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120222(US8691753, 71)
Affinity DataKi:  1.05nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120212(US8691753, 72 | US8691753, 61)
Affinity DataKi:  1.63nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120242(US8691753, 91)
Affinity DataKi:  1.84nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120246(US8691753, 96 | US8691753, 95)
Affinity DataKi:  1.92nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120191(US8691753, 39)
Affinity DataKi:  2.20nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120217(US8691753, 66)
Affinity DataKi:  2.20nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120252(US8691753, 101)
Affinity DataKi:  2.56nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120243(US8691753, 92)
Affinity DataKi:  2.58nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120254(US8691753, 103)
Affinity DataKi:  2.90nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120215(US8691753, 64)
Affinity DataKi:  3.30nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120168(US8691753, 16)
Affinity DataKi:  3.40nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120219(US8691753, 68)
Affinity DataKi:  3.5nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM92445(US8691753, 105 | Inhibitor, 10)
Affinity DataKi:  3.65nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM92443(US8691753, 97 | Thiophene derivative, compound 36 ...)
Affinity DataKi:  3.70nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120256(US8691753, 106)
Affinity DataKi:  4.30nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120221(US8691753, 70)
Affinity DataKi:  4.70nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120213(US8691753, 62)
Affinity DataKi:  5.20nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120173(US8691753, 21)
Affinity DataKi:  5.40nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120250(US8691753, 99)
Affinity DataKi:  5.40nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120216(US8691753, 65)
Affinity DataKi:  6.60nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetStromelysin-2(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120222(US8691753, 71)
Affinity DataKi:  7.70nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120220(US8691753, 69)
Affinity DataKi:  7.80nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120170(US8691753, 18)
Affinity DataKi:  8nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120241(US8691753, 90)
Affinity DataKi:  8nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120164(US8691753, 12)
Affinity DataKi:  8.20nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120155(US8691753, 3)
Affinity DataKi:  8.30nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120231(US8691753, 80)
Affinity DataKi:  8.60nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120157(US8691753, 5)
Affinity DataKi:  8.90nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120218(US8691753, 67)
Affinity DataKi:  10.2nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120222(US8691753, 71)
Affinity DataKi:  10.2nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120242(US8691753, 91)
Affinity DataKi:  10.3nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120225(US8691753, 74)
Affinity DataKi:  10.5nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120160(US8691753, 8)
Affinity DataKi:  11nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120175(US8691753, 23)
Affinity DataKi:  11.2nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120156(US8691753, 4)
Affinity DataKi:  11.8nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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Target72 kDa type IV collagenase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120221(US8691753, 70)
Affinity DataKi:  12nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120190(US8691753, 38)
Affinity DataKi:  12nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120203(US8691753, 52)
Affinity DataKi:  12.7nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120225(US8691753, 74)
Affinity DataKi:  13.5nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120234(US8691753, 83)
Affinity DataKi:  14.2nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120214(US8691753, 63)
Affinity DataKi:  14.3nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120251(US8691753, 100)
Affinity DataKi:  15.1nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetStromelysin-1(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120225(US8691753, 74)
Affinity DataKi:  16nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120238(US8691753, 87)
Affinity DataKi:  16.4nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120217(US8691753, 66)
Affinity DataKi:  16.4nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120219(US8691753, 68)
Affinity DataKi:  16.6nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetMacrophage metalloelastase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120244(US8691753, 93)
Affinity DataKi:  17nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetCollagenase 3(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120221(US8691753, 70)
Affinity DataKi:  17nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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TargetNeutrophil collagenase(Human)
French Alternative Energies and Atomic Energy Commission

US Patent
LigandPNGBDBM120241(US8691753, 90)
Affinity DataKi:  18nMAssay Description:The inhibition tests and the evaluation of the inhibition constants (Ki) on the various MMPs were carried out as described by Devel et al. (Devel et ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/6/2014
Entry Details
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