Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 6041
LigandPNGBDBM50403068(CHEMBL2216870 | IDELALISIB | US9745321, CAL-101)
Affinity DataIC50: 9nMAssay Description:Compounds of the invention were tested for inhibitory activity and potency against PI3Kδ.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2014
Entry Details
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PDB3D3D Structure (crystal)
LigandPNGBDBM104486(US8586597, 101 | USRE44599, 117)
Affinity DataIC50: 12nMAssay Description:Compounds of the invention were tested for inhibitory activity and potency against PI3Kδ.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2014
Entry Details
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LigandPNGBDBM104485(US8586597, 99 | USRE44599, 98)
Affinity DataIC50: 16nMAssay Description:Compounds of the invention were tested for inhibitory activity and potency against PI3Kδ.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2014
Entry Details
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LigandPNGBDBM104488(US8586597, 98 | USRE44599, 93)
Affinity DataIC50: 26nMAssay Description:Compounds of the invention were tested for inhibitory activity and potency against PI3Kδ.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2014
Entry Details
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LigandPNGBDBM104487(US8586597, 102 | USRE44599, 174)
Affinity DataIC50: 45nMAssay Description:Compounds of the invention were tested for inhibitory activity and potency against PI3Kδ.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2014
Entry Details
Go to US Patent