Compile Data Set for Download or QSAR
Report error Found 43 Enz. Inhib. hit(s) with all data for entry = 6023
TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104507(US8575114, III-2)
Affinity DataIC50: 11.4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104509(US8575114, III-4)
Affinity DataIC50: 23.6nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104500(US8575114, I-12)
Affinity DataIC50: 36.6nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104496(US8575114, I-8)
Affinity DataIC50: 81.1nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104489(US8575114, I-1)
Affinity DataIC50: 82.8nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104508(US8575114, III-3)
Affinity DataIC50: 83nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104492(US8575114, I-4)
Affinity DataIC50: 91nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104498(US8575114, I-10)
Affinity DataIC50: 94.8nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104497(US8575114, I-9)
Affinity DataIC50: 109nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104490(US8575114, I-2)
Affinity DataIC50: 129nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104494(US8575114, I-6)
Affinity DataIC50: 145nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104508(US8575114, III-3)
Affinity DataIC50: 148nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104502(US8575114, I-14)
Affinity DataIC50: 170nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104499(US8575114, I-11)
Affinity DataIC50: 222nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104501(US8575114, I-13)
Affinity DataIC50: 223nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104504(US8575114, II-1)
Affinity DataIC50: 226nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104491(US8575114, I-3)
Affinity DataIC50: 273nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104495(US8575114, I-7)
Affinity DataIC50: 316nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104506(US8575114, III-1)
Affinity DataIC50: 329nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104503(US8575114, I-15)
Affinity DataIC50: 463nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104510(US8575114, III-5)
Affinity DataIC50: 489nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104505(US8575114, II-2)
Affinity DataIC50: 542nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 2(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104493(US8575114, I-5)
Affinity DataIC50: 991nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104506(US8575114, III-1)
Affinity DataIC50: 6.25E+3nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104507(US8575114, III-2)
Affinity DataIC50: 1.75E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104489(US8575114, I-1)
Affinity DataIC50: 2.42E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104509(US8575114, III-4)
Affinity DataIC50: 3.54E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104498(US8575114, I-10)
Affinity DataIC50: 4.56E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104491(US8575114, I-3)
Affinity DataIC50: 4.95E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104496(US8575114, I-8)
Affinity DataIC50: 6.12E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104490(US8575114, I-2)
Affinity DataIC50: 6.74E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104505(US8575114, II-2)
Affinity DataIC50: 7.15E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104495(US8575114, I-7)
Affinity DataIC50: 7.32E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104510(US8575114, III-5)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104504(US8575114, II-1)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104503(US8575114, I-15)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104502(US8575114, I-14)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104501(US8575114, I-13)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
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TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104500(US8575114, I-12)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104497(US8575114, I-9)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104494(US8575114, I-6)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104493(US8575114, I-5)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent

TargetSodium/glucose cotransporter 1(Human)
Albany Molecular Research

US Patent
LigandPNGBDBM104492(US8575114, I-4)
Affinity DataIC50: 9.00E+4nMAssay Description:The inhibitory activity of the compounds of this invention against the SGLT-1 or SGLT-2 transporters.More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2014
Entry Details
Go to US Patent