Compile Data Set for Download or QSAR
Report error Found 42 Enz. Inhib. hit(s) with all data for entry = 5991
TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103737(US8563545, 11 | US10206907, Compound 234 | US11000...)
Affinity DataIC50: 7.69nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103737(US8563545, 11 | US10206907, Compound 234 | US11000...)
Affinity DataIC50: 15.5nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103736(US8563545, 10 | US10206907, Compound 207 | US11000...)
Affinity DataIC50: 18.2nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 31.4nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 38.7nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 41.2nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 47.1nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 48.3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 50.1nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 50.9nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 52.1nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 55.5nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
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TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 55.7nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103736(US8563545, 10 | US10206907, Compound 207 | US11000...)
Affinity DataIC50: 65.4nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 72.7nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 73.8nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 79.1nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 86.8nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103737(US8563545, 11 | US10206907, Compound 234 | US11000...)
Affinity DataIC50: 126nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 149nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 152nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 167nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 185nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 187nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 189nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103737(US8563545, 11 | US10206907, Compound 234 | US11000...)
Affinity DataIC50: 195nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103727(US8563545, 1 | US10112907, Example 00033 | US10206...)
Affinity DataIC50: 195nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103729(US8563545, 3 | US10206907, Compound 2 | US11000528...)
Affinity DataIC50: 291nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103735(US8563545, 9 | US10206907, Compound 141 | US110005...)
Affinity DataIC50: 334nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103734(US8563545, 8 | US10206907, Compound 140 | US110005...)
Affinity DataIC50: 435nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103733(US8563545, 7 | US10206907, Compound 139 | US110005...)
Affinity DataIC50: 504nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103735(US8563545, 9 | US10206907, Compound 141 | US110005...)
Affinity DataIC50: 849nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103730(US8563545, 4 | US10206907, Compound 6 | US11000528...)
Affinity DataIC50: 1.03E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103734(US8563545, 8 | US10206907, Compound 140 | US110005...)
Affinity DataIC50: 1.36E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103731(US8563545, 5 | US10206907, Compound 129 | US110005...)
Affinity DataIC50: 1.45E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103731(US8563545, 5 | US10206907, Compound 129 | US110005...)
Affinity DataIC50: 1.76E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetNon-receptor tyrosine-protein kinase TYK2(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 2.10E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK3(Human)
Galapagos

US Patent
LigandPNGBDBM103728(US8563545, 2 | US10206907, Compound 18 | US1100052...)
Affinity DataIC50: 2.84E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK1(Human)
Galapagos

US Patent
LigandPNGBDBM103732(US8563545, 6 | US10206907, Compound 130 | US110005...)
Affinity DataIC50: 3.45E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103732(US8563545, 6 | US10206907, Compound 130 | US110005...)
Affinity DataIC50: 5.07E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103733(US8563545, 7 | US10206907, Compound 139 | US110005...)
Affinity DataIC50: 6.45E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent

TargetTyrosine-protein kinase JAK2(Human)
Galapagos

US Patent
LigandPNGBDBM103734(US8563545, 8 | US10206907, Compound 140 | US110005...)
Affinity DataIC50: 7.73E+3nMAssay Description:In vitro inhibition assay using various enzyme.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2014
Entry Details
Go to US Patent