Compile Data Set for Download or QSAR
Report error Found 20 Enz. Inhib. hit(s) with all data for entry = 5904
TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25367((5R)-1,3-dioxepan-5-yl N-[(2S,3R)-3-hydroxy-4-[(4-...)
Affinity DataKi:  0.0260nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
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Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25371(US8501961, 22 | US8501961, 3h | 1,3-dioxan-5-yl N-...)
Affinity DataKi:  0.0410nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
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Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99910(US8501961, 102)
Affinity DataKi:  0.110nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99897(US8501961, 3a)
Affinity DataKi:  0.150nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99898(US8501961, 3b)
Affinity DataKi:  0.160nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99899(US8501961, 3c)
Affinity DataKi:  0.160nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99914(US8501961, 103)
Affinity DataKi:  0.180nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99916(US8501961, 130)
Affinity DataKi:  0.340nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99911(US8501961, 126)
Affinity DataKi:  0.400nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99915(US8501961, 129)
Affinity DataKi:  0.5nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99913(US8501961, 128)
Affinity DataKi:  0.510nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99902(US8501961, 3f)
Affinity DataKi:  0.740nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99901(US8501961, 3e)
Affinity DataKi:  0.810nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25375(4,4-dioxo-1,7,4-dioxathiecan-9-yl N-[(2S,3R)-3-hyd...)
Affinity DataKi:  1.90nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM99912(US8501961, 127)
Affinity DataKi:  5.40nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25374(US8501961, 25 | 1,3,6,10-tetraoxacyclododecan-8-yl...)
Affinity DataKi:  6.30nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25372(US8501961, 23 | 1,4,7-trioxecan-9-yl N-[(2S,3R)-3-...)
Affinity DataKi:  16nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25376(4-methyl-1,7,4-dioxazecan-9-yl N-[(2S,3R)-3-hydrox...)
Affinity DataKi:  19nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25370(US8501961, 21 | cycloheptyl N-[(2S,3R)-3-hydroxy-4...)
Affinity DataKi:  27nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
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TargetGag-Pol polyprotein(HIV-1)
Purdue Research Foundation

US Patent
LigandPNGBDBM25373(US8501961, 24 | 1,4,7,10-tetraoxacyclotridecan-12-...)
Affinity DataKi:  33nMAssay Description:Enzyme inhibitory assay utilizes a protocol described by Toth and Marshall (Toth, M. V.; Marshall G.R. A simple, continuous fluormetric assay for HIV...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/16/2013
Entry Details
Go to US Patent