Compile Data Set for Download or QSAR
Report error Found 32 Enz. Inhib. hit(s) with all data for entry = 12941
TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743229(Preparation of (S)-2-(6,8-dimethyl-4-oxopyrrolo[1,...)
Affinity DataEC50:  34nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743244(US20250163065, Compound I-46)
Affinity DataEC50:  68nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743243(Preparation of (S)-2 (6-methyl-4-oxopyrrolo[1,2-d]...)
Affinity DataEC50:  22nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743242(Preparation of (S)—N-(2-methyl-1-(4-trifluoromethy...)
Affinity DataEC50:  125nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743241(Preparation of (S)—N-(1-(4-fluorophenyl)-2-methylp...)
Affinity DataEC50:  26nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743240(Preparation of (S)—N-(2-methyl-1-(4-trifluoromethy...)
Affinity DataEC50:  61nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743239(Preparation of (S)—N-(1-(4-fluorophenyl)-2-methylp...)
Affinity DataEC50:  120nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743238(Preparation of (S)—N-(2-methyl-1-phenylpropyl)-2-(...)
Affinity DataEC50:  57nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743237(Preparation of (S)-2-(4-oxopyrrolo[1,2-d][1,2,4]tr...)
Affinity DataEC50:  61nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743236(Preparation of (S)—N-1-(4-bromophenyl)ethyl-2-(6-m...)
Affinity DataEC50:  15nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743235(Preparation of (S)-2-(6-methyl-4-oxopyrrolo[1,2-d]...)
Affinity DataEC50:  42nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743234(Preparation of (S)—N-(1-(4-bromophenyl)ethyl-2-(4-...)
Affinity DataEC50:  33nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743233(Preparation of (S)—N-(1-(naphthalen-1-ethyl)-2-(4-...)
Affinity DataEC50:  23nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743232(Preparation of (S)—N-1-(4-chlorophenyl)ethyl-2-(6,...)
Affinity DataEC50:  56nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743231(Preparation of (S)-2-(6,8-dimethyl-4-oxopyrrolo[1,...)
Affinity DataEC50:  96nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743230(Preparation of (S)-2-(6,8-dimethyl-4-oxopyrrolo[1,...)
Affinity DataEC50:  19nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM263368((s)-2-(4-oxobenzo[d][1,2,3]triazin-3(4h)-yl)-n-(1-...)
Affinity DataEC50:  61nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743228(Preparation of (S)-2-(6,8-dimethyl-4-oxopyrrolo[1,...)
Affinity DataEC50:  93nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743227(Preparation of (S)-2-(6,8-dimethyl-4-oxopyrrolo[1,...)
Affinity DataEC50:  95nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743226(Preparation of (S)—N-1-(4-chlorophenyl)ethyl-2-(6-...)
Affinity DataEC50:  23nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743225(Preparation of (S)-2-(6-methyl-4-oxopyrrolo[1,2-d]...)
Affinity DataEC50:  75nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743224(Preparation of (S)-2-(6-methyl-4-oxopyrrolo[1,2-d]...)
Affinity DataEC50:  13nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743223(Preparation of (S)—N-(1-(4-methoxyphenyl)ethyl-2-(...)
Affinity DataEC50:  24nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743222(Preparation of (S)-2-(6-methyl-4-oxopyrrolo[1,2-d]...)
Affinity DataEC50:  21nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743221(Preparation of (S)—N-(1-(4-fluorophenyl)ethyl-2-(6...)
Affinity DataEC50:  19nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743220(Preparation of (S)-2-(4-oxopyrrolo[1,2-d][1,2,4]tr...)
Affinity DataEC50:  45nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743219(Preparation of (S)—N-1-(4-chlorophenyl)ethyl-2-(4-...)
Affinity DataEC50:  30nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743218(Preparation of (S)-2-(4-oxopyrrolo[1,2-d][1,2,4]tr...)
Affinity DataEC50:  25nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743217(Preparation of (S)-2-(4-oxopyrrolo[1,2-d][1,2,4]tr...)
Affinity DataEC50:  111nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743216(Preparation of (S)—N-(1-(4-methoxyphenyl)ethyl)-2-...)
Affinity DataEC50:  60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743215(Preparation of (S)-2-(4-oxopyrrolo[1,2-d][1,2,4]tr...)
Affinity DataEC50:  28nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

TargetProbable G-protein coupled receptor 139(Human)
Shanghaitech University

US Patent
LigandPNGBDBM743214(Preparation of (S)—N-(1-(4-fluorophenyl)ethyl-2-(4...)
Affinity DataEC50:  56nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent