Compile Data Set for Download or QSAR
Report error Found 142 Enz. Inhib. hit(s) with all data for entry = 12940
Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743171(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743171(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Affinity DataIC50: 0.800nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743142(US20250163064, Example 1)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743142(US20250163064, Example 1)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743172(2-Amino-4-(4- (azocan-1-yl)-6- chloro-8-fluoro- 2-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
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Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743172(2-Amino-4-(4- (azocan-1-yl)-6- chloro-8-fluoro- 2-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
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Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743194((2S)-1-(7-(2- Amino-3-cyano- 7- fluorobenzo[b] thi...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
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Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743194((2S)-1-(7-(2- Amino-3-cyano- 7- fluorobenzo[b] thi...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743199(2-Amino-4-(6- chloro-8-fluoro- 4-(6-fluoro-1,4- ox...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743203(US20250163064, Example 62)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743149(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743157(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7a.S)-2- fl...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743159(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743159(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743163(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743163(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743165(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743168(2-Amino-4-(6- chloro-8-fluoro- 4-(3- fluoroazepan-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743168(2-Amino-4-(6- chloro-8-fluoro- 4-(3- fluoroazepan-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743173(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743173(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743185(2-Amino-4-(6- chloro-4-(6- ethyl-6-hydroxy- 1,4-ox...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743192(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743192(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743200(2-Amino-4-(6- chloro-8-fluoro- 4-(6-fluoro-1,4- ox...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743146(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7a.S)-2- fl...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743156(1-(7-(2-Amino-3- cyano-7- fluorobenzo[b] thiophen-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743157(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7a.S)-2- fl...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743158(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743165(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743166(2-Amino-4-(6- chloro-4-(1,1- dioxido-1,4- thiazepa...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743166(2-Amino-4-(6- chloro-4-(1,1- dioxido-1,4- thiazepa...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743169(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743174(4-(4-(6-Oxa-3- azabicyclo[3.2.1] octan-3-yl)-6- ch...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743174(4-(4-(6-Oxa-3- azabicyclo[3.2.1] octan-3-yl)-6- ch...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743182(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743185(2-Amino-4-(6- chloro-4-(6- ethyl-6-hydroxy- 1,4-ox...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743187(2-Amino-4-(6- chloro-4-(6- (difluoromethyl)- 6-hyd...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743198(1-(7-(2-Amino-3- cyano-7- fluorobenzo[b] thiophen-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743198(1-(7-(2-Amino-3- cyano-7- fluorobenzo[b] thiophen-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743199(2-Amino-4-(6- chloro-8-fluoro- 4-(6-fluoro-1,4- ox...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743202(US20250163064, Example 61)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743203(US20250163064, Example 62)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743204(US20250163064, Example 63)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743144(1-(7-(2-Amino-3- cyano-7- fluorobenzo[b] thiophen-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743145(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743146(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7a.S)-2- fl...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743148(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d coupled exchange(Human)
Amgen

US Patent
LigandPNGBDBM743149(2-Amino-4-(6- chloro-8-fluoro- 2-(((2R,7aS)-2- flu...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

Targetkras g12d tr-fret(Human)
Amgen

US Patent
LigandPNGBDBM743155(chloro-8-fluoro- 2-(((2R,7aS)-2- fluorotetrahydro-...)
Ligand Info
In Depth
Date in BDB:
9/19/2025
Entry Details
Go to US Patent

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