Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 12905
TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662989(Synthesis of N-(5-((1H-pyrazol-1-yl)methyl)-3,4-di...)
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739500(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.300nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739493(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.400nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662990(Synthesis of N-(5-((1H-pyrazol-1-yl)methyl)-3,4-di...)
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739494(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662985(Synthesis of 7-chloro-1-(2-chlorophenyl)-4-(prop-2...)
Affinity DataIC50: 0.600nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739495(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739496(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6B(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662989(Synthesis of N-(5-((1H-pyrazol-1-yl)methyl)-3,4-di...)
Affinity DataIC50: 0.700nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739497(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 0.900nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739492(N-(4-((1H-pyrazol-1-yl)methyl)-2,2-difluoro-[1,3]d...)
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6B(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662985(Synthesis of 7-chloro-1-(2-chlorophenyl)-4-(prop-2...)
Affinity DataIC50: 1.10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM722767(US20250059204, Compound 44 | US20250145637, Exampl...)
Affinity DataIC50: 1.20nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6B(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM662990(Synthesis of N-(5-((1H-pyrazol-1-yl)methyl)-3,4-di...)
Affinity DataIC50: 1.40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6B(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739492(N-(4-((1H-pyrazol-1-yl)methyl)-2,2-difluoro-[1,3]d...)
Affinity DataIC50: 1.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739498(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 1.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739502(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 1.90nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM722787(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 2.70nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM722778(US20250059204, Compound 55 | US20250145637, Exampl...)
Affinity DataIC50: 2.90nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739491(N-(5-((1H-pyrazol-1-yl)methyl)-2,3-dihydro-[1,4]di...)
Affinity DataIC50: 4.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739507(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 4.60nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739508(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 4.70nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739509(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 4.80nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739511((R)-2,6-dimethoxy-N-(4-(tetrahydrofuran-2-yl)-2,3-...)
Affinity DataIC50: 5.20nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739503(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 10.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739510(2,6-dimethoxy-N-(4-(tetrahydrofuran-2-yl)-2,3-dihy...)
Affinity DataIC50: 12.2nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739504(N-(4-((1H-pyrazol-1-yl)methyl)-2,3-dihydrobenzofur...)
Affinity DataIC50: 12.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent

TargetHistone acetyltransferase KAT6A(Human)
Jiangsu Hengrui Pharmaceuticals

US Patent
LigandPNGBDBM739499(N-(5-((1H-pyrazol-1-yl)methyl)-3,4-dihydro-2H-chro...)
Affinity DataIC50: 12.5nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
9/9/2025
Entry Details
Go to US Patent