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Found
29
Enz. Inhib. hit(s) with all data for entry = 12842
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732865
(2-(4,4-difluoroazepan-1-yl)-6,7-difluoro-N-(3-sulf...)
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Affinity Data
IC50: 0.0710nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732865
(2-(4,4-difluoroazepan-1-yl)-6,7-difluoro-N-(3-sulf...)
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Affinity Data
IC50: 0.0840nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732866
(2-(4,4-difluoroazepan-1-yl)-6,7-difluoro-N-(2-sulf...)
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Affinity Data
IC50: 0.0950nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732864
(2-(4,4-difluoroazepan-1-yl)-N-(2-sulfamoylpyridine...)
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Affinity Data
IC50: 0.340nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732867
(N-(3-carbamoyl-4-fluorophenyl)-2-(4,4-difluoroazep...)
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Affinity Data
IC50: 0.360nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732863
(N-(2-carbamoylpyridin-4-yl)-2-(4,4-difluoroazepan-...)
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Affinity Data
IC50: 0.460nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732864
(2-(4,4-difluoroazepan-1-yl)-N-(2-sulfamoylpyridine...)
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Affinity Data
IC50: 0.725nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732863
(N-(2-carbamoylpyridin-4-yl)-2-(4,4-difluoroazepan-...)
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Affinity Data
IC50: 0.784nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732862
(US20250115578, KH09 | US20250115578, Example 09)
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Affinity Data
IC50: 0.918nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732862
(US20250115578, KH09 | US20250115578, Example 09)
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Affinity Data
IC50: 1nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732869
(N-(2-carbamoylpyridin-4-yl)-2-(4,4-difluoroazepan-...)
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Affinity Data
IC50: 1.5nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732861
(US20250115578, KH08 | US20250115578, Example 08)
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Affinity Data
IC50: 1.74nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732854
(US20250115578, KH02 | US20250115578, Example 02)
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Affinity Data
IC50: 2.82nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732859
(US20250115578, KH06 | US20250115578, Example 06)
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Affinity Data
IC50: 3.10nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732861
(US20250115578, KH08 | US20250115578, Example 08)
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Affinity Data
IC50: 3.30nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732854
(US20250115578, KH02 | US20250115578, Example 02)
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Affinity Data
IC50: 5.30nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732872
(2-(4,4-difluoroazepan-1-yl)-N-(2-(S-methylsulfonim...)
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Affinity Data
IC50: 8nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732858
(US20250115578, KH05 | US20250115578, Example 05)
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Affinity Data
IC50: 8.90nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732871
(N-(2-carbamoylpyridin-4-yl)-2-(4,4-difluoroazepan-...)
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Affinity Data
IC50: 9.23nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM181223
(US9139529, 66 | US9783501, Compound 66 | US2025011...)
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Affinity Data
IC50: 9.5nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732855
(US20250115578, KH03 | US20250115578, Example 03)
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Affinity Data
IC50: 10nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732873
(2-(4,4-difluoroazepan-1-yl)-N-(2-(N-methylsulfamoy...)
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Affinity Data
IC50: 11.4nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732860
(US20250115578, KH07 | US20250115578, Example 07)
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Affinity Data
IC50: 14.7nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
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Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM161225
(US9163042, 9a | US9051270, 10 | US10087143, Compou...)
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Affinity Data
IC50: 16nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
Copy Rxn URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732858
(US20250115578, KH05 | US20250115578, Example 05)
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Affinity Data
IC50: 21.3nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
Copy Rxn URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM161225
(US9163042, 9a | US9051270, 10 | US10087143, Compou...)
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Affinity Data
IC50: 35.1nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
Copy Rxn URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732857
(US20250115578, KH04 | US20250115578, Example 04)
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Affinity Data
IC50: 66.7nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
Copy Rxn URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732870
(N-(2-carbamoylpyridin-4-yl)-2-(4,4-difluoroazepan-...)
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Affinity Data
IC50: 97.1nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
Go to US Patent
Copy Rxn URL
Target
Sodium channel protein type 10 subunit alpha
(Human)
Chengdu Kanghong Pharmaceutical
US Patent
Ligand
BDBM732853
(US20250115578, KH01 | US20250115578, Example 01)
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Affinity Data
IC50: 100nM
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Date in BDB:
8/22/2025
Entry Details
Copy Entry DOI
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BDBM161225
