Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 12715
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722401((E)-1-(2-(2-(mesitylimino)-10-methoxy-9-(methoxy-d...)
Affinity DataIC50: 50nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
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TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722421((E)-1-(2-(2-((4-cyclopropyl-2,6-dimethylphenyl)imi...)
Affinity DataIC50: 50nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722427((E)-1-(2-(9-ethoxy-2-(mesitylimino)-10-methoxy-4-o...)
Affinity DataIC50: 50nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722436((E)-1-(2-(2-(mesitylimino)-9-methoxy-10-(methoxy-d...)
Affinity DataIC50: 50nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722405((E)-1-(2-(2-((2,6-dimethyl-4-(trifluoromethyl)phen...)
Affinity DataIC50: 75nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Xizang Haisco Pharmaceutical

US Patent
LigandPNGBDBM722429((E)-1-(2-(2-((4-fluoro-2,6-dimethylphenyl)imino)-9...)
Affinity DataIC50: 75nMAssay Description:1) Prepare FAM cAMP working solution: 20 μL of FAM-Cyclic-3′, 5′-AMP stock was added to 1980 μL of PDE assay buffer. The mixture was added to all wel...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/19/2025
Entry Details
Go to US Patent