Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 12675
TargetRelaxin receptor 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM719052(6-fluoro-3'-(((1S,5R,6S,7R)-7-((4-fluoro-3-(triflu...)
Affinity DataEC50:  1.19E+3nMAssay Description:Human embryonic kidney cells 293 (HEK293) cells and HEK293 cells stably expressing human RXFP1, were cultured in MEM medium supplemented with 10% qua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
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TargetRelaxin receptor 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM719069((1R,5S,6R,7S)-N- (4-fluoro-3-(tri- fluoromethyl)- ...)
Affinity DataEC50:  823nMAssay Description:Human embryonic kidney cells 293 (HEK293) cells and HEK293 cells stably expressing human RXFP1, were cultured in MEM medium supplemented with 10% qua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
Go to US Patent

TargetRelaxin receptor 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM719070((1R,5S,6R,7S)-N- (4-fluoro-3-(tri- fluoromethyl)- ...)
Affinity DataEC50:  916nMAssay Description:Human embryonic kidney cells 293 (HEK293) cells and HEK293 cells stably expressing human RXFP1, were cultured in MEM medium supplemented with 10% qua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
Go to US Patent

TargetRelaxin receptor 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM719071((1R,5S,6R,7S)-N- (4-fluoro-3-(tri- fluoromethyl)- ...)
Affinity DataEC50:  2.23E+3nMAssay Description:Human embryonic kidney cells 293 (HEK293) cells and HEK293 cells stably expressing human RXFP1, were cultured in MEM medium supplemented with 10% qua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
Go to US Patent

TargetRelaxin receptor 1(Human)
Bristol-Myers Squibb

US Patent
LigandPNGBDBM719072(2-(6-fluoro-3'-(((1S,5R,6S,7R)-7-((4-fluoro-3-(tri...)
Affinity DataEC50:  12nMAssay Description:Human embryonic kidney cells 293 (HEK293) cells and HEK293 cells stably expressing human RXFP1, were cultured in MEM medium supplemented with 10% qua...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/16/2025
Entry Details
Go to US Patent