Compile Data Set for Download or QSAR
Report error Found 39 Enz. Inhib. hit(s) with all data for entry = 12617
TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714736(US20250026742, Example 35-1)
Affinity DataIC50: 0.410nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714737(5-(5-amino-6-(5-(4-((1-methylpiperidin-4-yl)amino)...)
Affinity DataIC50: 0.570nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714724(1-(4-(5-(3-amino-6-(4-(cyclopropylsulfonyl)phenyl)...)
Affinity DataIC50: 0.700nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714728(1-(4-(5-(3-amino)-6-(1,1-dioxo-2,3-dihydrobenzo[b]...)
Affinity DataIC50: 0.75nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714739(US20250026742, Example 38-1)
Affinity DataIC50: 0.75nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714738(5-(5-amino-6-(5-(4-((methylamino)methyl)phenyl)-1,...)
Affinity DataIC50: 0.770nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714712(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 0.820nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714705(1-(4-(5-(3-amino-6-(4-isopropylsulfonyl)phenyl)pyr...)
Affinity DataIC50: 0.830nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714734(US20250026742, Example 33-1)
Affinity DataIC50: 0.830nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714735(5-(5-amino-6-(5-(4-((methylamino)methyl)phenyl)iso...)
Affinity DataIC50: 0.920nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714718(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 0.930nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714664(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 0.970nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714708(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.04nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714725(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.08nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714719(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.16nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714723(5-(5-(3-amino-6-(4-(propan-2-ylsulfonimido)phenyl)...)
Affinity DataIC50: 1.21nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714720(1-(6-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.26nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714729(N-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.29nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714722(5-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)pyraz...)
Affinity DataIC50: 1.31nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714715(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.42nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714704(US20250026742, Example 3)
Affinity DataIC50: 1.60nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714714(1-(4-(5-(3-amino-6-(4-(N-methylpropan-2-yl-sulfoni...)
Affinity DataIC50: 1.68nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714711(4-(5-amino-6-(3-(4-(guanidinomethyl)phenyl)isoxazo...)
Affinity DataIC50: 1.75nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714721(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 1.81nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714710(US20250026742, Example 9)
Affinity DataIC50: 1.83nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM50226746(Berzosertib | VX-970 | US20250026742, Example VX-9...)
Affinity DataIC50: 1.94nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714726(4-(5-amino-6-(3-(4-(guanidinomethyl)phenyl)isoxazo...)
Affinity DataIC50: 1.98nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714716(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 2nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714727(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)pyraz...)
Affinity DataIC50: 2.06nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714733(5-(5-amino-6-(3-(4-((methylamino)methyl)phenyl)iso...)
Affinity DataIC50: 2.09nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714706(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 2.32nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714713(1-(4-(5-(3-amino-6-(4-(N,S-dimethylsulfonylimino)p...)
Affinity DataIC50: 2.53nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714703((4-(5-amino-6-(3-(4-((methylamino)methyl)phenyl)is...)
Affinity DataIC50: 2.79nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714707(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 2.90nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714730(N-(4-(5-(3-Amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 3.12nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714731(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 3.35nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714709(3-(3-(4-((aminosulfonyl)aminomethylene)phenyl)isox...)
Affinity DataIC50: 3.64nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714732(5-(5-(3-amino-6-(4-isopropylsulfonyl)phenyl)pyrazi...)
Affinity DataIC50: 4nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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TargetSerine/threonine-protein kinase ATR(Human)
Suzhou Ark Biopharmaceutical Co.

US Patent
LigandPNGBDBM714717(1-(4-(5-(3-amino-6-(4-(isopropylsulfonyl)phenyl)py...)
Affinity DataIC50: 9.74nMAssay Description:Prepare various buffer systems required for the experiment:1. Prepare ATR reaction buffer containing 25 mM HEPES (Gibco, Cat #15630-080), 5 mM DTT (S...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/30/2025
Entry Details
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