Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 12569
TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710426(US20250002435, Compound HU-308)
Affinity DataKi:  1.16nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
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TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710405(US20250002435, Compound 1d)
Affinity DataKi:  3.51nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710423(US20250002435, Compound 5b)
Affinity DataKi: >10nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710422(US20250002435, Compound 5a)
Affinity DataKi: >10nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710403(US20250002435, Compound 1b)
Affinity DataKi:  14.4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710425(US20250002435, Compound 5d)
Affinity DataKi:  24.6nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710419(US20250002435, Compound 4b)
Affinity DataKi:  28.3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710423(US20250002435, Compound 5b)
Affinity DataKi:  36.5nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710399(US20250002435, Compound 1a)
Affinity DataKi:  47.7nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710421(US20250002435, Compound 4d)
Affinity DataKi:  56.6nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710404(US20250002435, Compound 1c)
Affinity DataKi:  56.8nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710409(US20250002435, Compound 2b)
Affinity DataKi:  73.4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710424(US20250002435, Compound 5c)
Affinity DataKi:  107nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710418(US20250002435, Compound 4a)
Affinity DataKi:  155nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710408(US20250002435, Compound 2a)
Affinity DataKi:  224nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710407(US20250002435, Compound 1f)
Affinity DataKi:  233nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710405(US20250002435, Compound 1d)
Affinity DataKi:  427nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710420(US20250002435, Compound 4c)
Affinity DataKi:  438nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710412(US20250002435, Compound 3c)
Affinity DataKi:  444nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710425(US20250002435, Compound 5d)
Affinity DataKi:  451nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710417(US20250002435, Compound 3h)
Affinity DataKi:  494nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710411(US20250002435, Compound 3b)
Affinity DataKi:  610nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710413(US20250002435, Compound 3d)
Affinity DataKi:  834nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710410(US20250002435, Compound 3a)
Affinity DataKi:  1.01E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710415(US20250002435, Compound 3f)
Affinity DataKi:  1.45E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710416(US20250002435, Compound 3g)
Affinity DataKi:  1.65E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710403(US20250002435, Compound 1b)
Affinity DataKi:  2.29E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710414(US20250002435, Compound 3e)
Affinity DataKi:  2.87E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710422(US20250002435, Compound 5a)
Affinity DataKi:  4.98E+3nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710399(US20250002435, Compound 1a)
Affinity DataKi: >1.00E+4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 2(Human)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710406(US20250002435, Compound 1e)
Affinity DataKi: >1.00E+4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710419(US20250002435, Compound 4b)
Affinity DataKi: >1.00E+4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710418(US20250002435, Compound 4a)
Affinity DataKi: >1.00E+4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent

TargetCannabinoid receptor 1(Mouse)
Hebrew University of Jerusalem

US Patent
LigandPNGBDBM710409(US20250002435, Compound 2b)
Affinity DataKi: >1.00E+4nMAssay Description:Binding to the CB1R was assessed in a competition displacement assays using [3H]CP-55,940 as the radioligand and crude membranes from mouse brain for...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/15/2025
Entry Details
Go to US Patent