Compile Data Set for Download or QSAR
Report error Found 54 Enz. Inhib. hit(s) with all data for entry = 12506
TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707203((R)-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyri...)
Affinity DataIC50: 0.290nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707205((S)-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyri...)
Affinity DataIC50: 0.310nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707204((S)-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyri...)
Affinity DataIC50: 0.320nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707191(N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyrid...)
Affinity DataIC50: 0.320nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707202((R)-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyri...)
Affinity DataIC50: 0.330nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707230(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.350nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707201(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.350nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707213(7-((4-(6-(1H-pyrazol-5-yl)pyridin-3-yl)piperazin-1...)
Affinity DataIC50: 0.450nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707212(7-((4-(6-(1H-1,2,3-triazol-5-yl)pyridin-3-yl)piper...)
Affinity DataIC50: 0.450nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707210(N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyrid...)
Affinity DataIC50: 0.480nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707206(N-(azetidin-3-yl)-5-(4-((7-ethyl-6-oxo-5,6-dihydro...)
Affinity DataIC50: 0.510nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707200(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.510nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707195(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.540nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707194(N-cyclobutyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-...)
Affinity DataIC50: 0.560nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707229(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.560nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707190(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.560nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707219((S)—N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphth...)
Affinity DataIC50: 0.580nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707192(methyl(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphth...)
Affinity DataIC50: 0.580nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707223(N-(cyclopropylmethyl)-5-(4-((7-ethyl-6-oxo-5,6-dih...)
Affinity DataIC50: 0.610nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707199(3-ethyl-7-((4-(2-methylimidazo[1,2-a]pyrazin-6-yl)...)
Affinity DataIC50: 0.650nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707217((1R,2R)—N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-na...)
Affinity DataIC50: 0.660nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707232(US20240400586, Compound 51)
Affinity DataIC50: 0.660nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707207(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.670nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707225(3-ethyl-7-((4-(6-(5-methyl-4H-1,2,4-triazol-3-yl)p...)
Affinity DataIC50: 0.670nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707189(N-cyclopropyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5...)
Affinity DataIC50: 0.670nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707231(US20240400586, Compound 50)
Affinity DataIC50: 0.690nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707221(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.700nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707198(1-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyrid...)
Affinity DataIC50: 0.710nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707193(N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyrid...)
Affinity DataIC50: 0.730nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707228(2 (1H)-one | US20240400586, Compound 45)
Affinity DataIC50: 0.730nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707208(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.730nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707216(N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyrid...)
Affinity DataIC50: 0.740nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707211(3-ethyl-7-((4-(2-methylimidazo[1,2-b]pyridazin-6-y...)
Affinity DataIC50: 0.75nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707197(N-cyclopropyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5...)
Affinity DataIC50: 0.760nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707222(N-(bicyclo[1.1.1]pentan-1-yl)-5-(4-((7-ethyl-6-oxo...)
Affinity DataIC50: 0.770nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707224(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 0.840nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707209(N-(3,3-difluorocyclobutyl)-5-(4-((7-ethyl-6-oxo-5,...)
Affinity DataIC50: 0.880nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707227(3-ethyl-7-((4-(2-ethylimidazo[1,2-a]pyrazin-6-yl)p...)
Affinity DataIC50: 0.920nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707226(3-ethyl-7-((4-(2-(trifluoromethyl)imidazo[1,2-a]py...)
Affinity DataIC50: 0.930nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707220(Cyclopropyl(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-n...)
Affinity DataIC50: 0.960nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707218((1S,2R)—N-(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-na...)
Affinity DataIC50: 0.970nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707188(3-ethyl-7-((4-(6-(5-methyl-1,3,4-oxadiazol-2-yl)py...)
Affinity DataIC50: 1.33nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707196(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 1.60nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707214(3-ethyl-7-((4-(2-methyl-[1,2,4]triazolo[1,5-a]pyri...)
Affinity DataIC50: 1.70nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707215(3-ethyl-7-((4-(6-((1-methyl-1H-pyrazol-3-yl)amino)...)
Affinity DataIC50: 2nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707187(5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5-naphthyridin-...)
Affinity DataIC50: 2.01nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 1(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707186(3-ethyl-7-((4-(2-methyl-1-oxoisoindolin-5-yl)piper...)
Affinity DataIC50: 3.66nMAssay Description:Table 1: PARP1 chemical fluorescence detection kit was purchased from BPS Bioscience. The histone solution in the kit was diluted 5× with 1×PBS, and ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase 2(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707189(N-cyclopropyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5...)
Affinity DataIC50: 27.5nMAssay Description:Table 2: PARP2, PARP5A, PARP5B, PARP6, PARP7, PARP14 and PARP15 chemical fluorescence detection kits were purchased from BPS Bioscience. The histone ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetPoly [ADP-ribose] polymerase tankyrase-2(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707189(N-cyclopropyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5...)
Affinity DataIC50: 576nMAssay Description:Table 2: PARP2, PARP5A, PARP5B, PARP6, PARP7, PARP14 and PARP15 chemical fluorescence detection kits were purchased from BPS Bioscience. The histone ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetProtein mono-ADP-ribosyltransferase PARP15(Human)
Haisco Pharmaceutical Group

US Patent
LigandPNGBDBM707189(N-cyclopropyl-5-(4-((7-ethyl-6-oxo-5,6-dihydro-1,5...)
Affinity DataIC50: 4.30E+3nMAssay Description:Table 2: PARP2, PARP5A, PARP5B, PARP6, PARP7, PARP14 and PARP15 chemical fluorescence detection kits were purchased from BPS Bioscience. The histone ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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