Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 12496
TargetAcetyl-CoA carboxylase 2(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM50189617({(3R)-1'-(anthracen-9-ylcarbonyl)[1,4'-bipiperidin...)
Affinity DataIC50: 78.1nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetATP-citrate synthase(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM50209010(3,5-dichloro-2-hydroxy-N-(4-methoxy-biphenyl-3-yl)...)
Affinity DataIC50: 445nMAssay Description:Table 4: ATP citrate lyase was obtained from Sino Biological Inc. Cat #11769-H07B, Lot #LC08DE1701. It was prepared from a DNA sequence encoding the ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetATP-citrate synthase(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706749(US20240398737, Compound I-32-CoA)
Affinity DataIC50: 988nMAssay Description:Table 4: ATP citrate lyase was obtained from Sino Biological Inc. Cat #11769-H07B, Lot #LC08DE1701. It was prepared from a DNA sequence encoding the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetAcetyl-CoA carboxylase 1(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM50189617({(3R)-1'-(anthracen-9-ylcarbonyl)[1,4'-bipiperidin...)
Affinity DataIC50: 2.14E+3nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/16/2025
Entry Details
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TargetATP-citrate synthase(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706750(US20240398737, Compound I-1-CoA)
Affinity DataIC50: 3.34E+3nMAssay Description:Table 4: ATP citrate lyase was obtained from Sino Biological Inc. Cat #11769-H07B, Lot #LC08DE1701. It was prepared from a DNA sequence encoding the ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetAcetyl-CoA carboxylase 2(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706749(US20240398737, Compound I-32-CoA)
Affinity DataIC50: 5.02E+3nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetAcetyl-CoA carboxylase 1(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706749(US20240398737, Compound I-32-CoA)
Affinity DataIC50: 5.07E+3nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetAcetyl-CoA carboxylase 2(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706750(US20240398737, Compound I-1-CoA)
Affinity DataIC50: 9.41E+3nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetAcetyl-CoA carboxylase 1(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706750(US20240398737, Compound I-1-CoA)
Affinity DataIC50: 1.63E+4nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent

TargetAcetyl-CoA carboxylase 1(Human)
Espervita Therapeutics

US Patent
LigandPNGBDBM706748(US20240398737, Compound I-32)
Affinity DataIC50: 2.84E+5nMAssay Description:Table 3: Human ACC1 (Cat #50202 Lot #120830) and ACC2 (Cat #50201 Lot #160217) were obtained from BPS Biosciences, San Diego, CA 92121. Human ACC1 ha...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/16/2025
Entry Details
Go to US Patent