Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 12442
TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702990(US20240366807, Compound 3860-BD-B)
Affinity DataIC50: 0.400nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702991(US20240366807, Compound 7290B)
Affinity DataIC50: 13.9nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM50431239(CHEMBL2333029 | US20240366807, Formula I.7)
Affinity DataIC50: 14nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM50431239(CHEMBL2333029 | US20240366807, Formula I.7)
Affinity DataIC50: 15nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM50431237(CHEMBL2332617 | US20240366807, Formula I.8)
Affinity DataIC50: 15.6nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM50431237(CHEMBL2332617 | US20240366807, Formula I.8)
Affinity DataIC50: 16.7nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702984(US20240366807, Formula I.6)
Affinity DataIC50: 48nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702984(US20240366807, Formula I.6)
Affinity DataIC50: 53nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702988(US20240366807, Formula I.10)
Affinity DataIC50: 100nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702989(US20240366807, Formula I.11)
Affinity DataIC50: 130nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702988(US20240366807, Formula I.10)
Affinity DataIC50: 130nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702984(US20240366807, Formula I.6)
Affinity DataIC50: 130nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702984(US20240366807, Formula I.6)
Affinity DataIC50: 130nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702987(US20240366807, Formula I.9)
Affinity DataIC50: 140nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702987(US20240366807, Formula I.9)
Affinity DataIC50: 140nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702989(US20240366807, Formula I.11)
Affinity DataIC50: 150nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702975(US20240366807, Formula I.1)
Affinity DataIC50: 220nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702983(US20240366807, Formula I.5)
Affinity DataIC50: 240nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702983(US20240366807, Formula I.5)
Affinity DataIC50: 240nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702975(US20240366807, Formula I.1)
Affinity DataIC50: 260nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702982(US20240366807, Formula I.4)
Affinity DataIC50: 330nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702981(US20240366807, Formula I.3)
Affinity DataIC50: 390nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702980(US20240366807, Formula I.2)
Affinity DataIC50: 390nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702982(US20240366807, Formula I.4)
Affinity DataIC50: 450nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702980(US20240366807, Formula I.2)
Affinity DataIC50: 650nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetProlyl endopeptidase FAP(Human)
Tufts College

US Patent
LigandPNGBDBM702981(US20240366807, Formula I.3)
Affinity DataIC50: 690nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702981(US20240366807, Formula I.3)
Affinity DataIC50: 790nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702982(US20240366807, Formula I.4)
Affinity DataIC50: 1.20E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM50431239(CHEMBL2333029 | US20240366807, Formula I.7)
Affinity DataIC50: 1.34E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702981(US20240366807, Formula I.3)
Affinity DataIC50: 1.40E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702982(US20240366807, Formula I.4)
Affinity DataIC50: 1.50E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM50431239(CHEMBL2333029 | US20240366807, Formula I.7)
Affinity DataIC50: 1.57E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702983(US20240366807, Formula I.5)
Affinity DataIC50: 1.90E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702989(US20240366807, Formula I.11)
Affinity DataIC50: 1.90E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702987(US20240366807, Formula I.9)
Affinity DataIC50: 2.00E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702983(US20240366807, Formula I.5)
Affinity DataIC50: 2.00E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM50431237(CHEMBL2332617 | US20240366807, Formula I.8)
Affinity DataIC50: 2.11E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702989(US20240366807, Formula I.11)
Affinity DataIC50: 2.20E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702980(US20240366807, Formula I.2)
Affinity DataIC50: 2.20E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702987(US20240366807, Formula I.9)
Affinity DataIC50: 2.30E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702988(US20240366807, Formula I.10)
Affinity DataIC50: 2.30E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent

TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM50431237(CHEMBL2332617 | US20240366807, Formula I.8)
Affinity DataIC50: 2.34E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702988(US20240366807, Formula I.10)
Affinity DataIC50: 2.50E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702980(US20240366807, Formula I.2)
Affinity DataIC50: 3.10E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702975(US20240366807, Formula I.1)
Affinity DataIC50: 4.10E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
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TargetPresequence protease, mitochondrial(Human)
Tufts College

US Patent
LigandPNGBDBM702975(US20240366807, Formula I.1)
Affinity DataIC50: 5.70E+3nMAssay Description:Enzymatic activity of DPPIV, DPP8, DPP9, FAP, and PREP was measured at 25° C. on a Molecular Devices M2e multidetection microtiter plate reader, moni...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/14/2025
Entry Details
Go to US Patent