Compile Data Set for Download or QSAR
Report error Found 3 Enz. Inhib. hit(s) with all data for entry = 12421
Target5-hydroxytryptamine receptor 2B(Human)
H. Lundbeck

US Patent
LigandPNGBDBM50373192(CHEMBL405519 | US10729710, Compound (I) | US202403...)
Affinity DataEC50:  2.90E+3nMAssay Description:Evaluation of the affinity of compounds for the human 5-HT2B receptor was determined in a radioligand binding assay at Eurofins/Cerep (France). Membr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2025
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2B(Human)
H. Lundbeck

US Patent
LigandPNGBDBM453276(US10729710, Compound (Ia) | US20240352055, Compoun...)
Affinity DataEC50: >6.00E+3nMAssay Description:Evaluation of the affinity of compounds for the human 5-HT2B receptor was determined in a radioligand binding assay at Eurofins/Cerep (France). Membr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2025
Entry Details
Go to US Patent

Target5-hydroxytryptamine receptor 2B(Human)
H. Lundbeck

US Patent
LigandPNGBDBM453277(US10729710, Compound (Ib) | US20240352055, Compoun...)
Affinity DataEC50:  3.80nMAssay Description:Evaluation of the affinity of compounds for the human 5-HT2B receptor was determined in a radioligand binding assay at Eurofins/Cerep (France). Membr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2025
Entry Details
Go to US Patent