Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 12363
TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698744(US20240317732, Compound XL5)
Affinity DataKd:  1.48E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698745(US20240317732, Compound XL23)
Affinity DataKd:  3.88E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
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TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698746(US20240317732, Compound XL24)
Affinity DataKd:  1.74E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698747(US20240317732, Compound XL25)
Affinity DataKd:  4.12E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698748(US20240317732, Compound XL26)
Affinity DataKd:  6.67E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698749(US20240317732, Compound XL27)
Affinity DataKd:  3.94E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698750(US20240317732, Compound XL28)
Affinity DataKd:  3.82E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698751(US20240317732, Compound XL29)
Affinity DataKd:  7.81E+3nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent

TargetProteasomal ubiquitin receptor ADRM1(Homo sapiens)
Department of Health And Human Service

US Patent
LigandPNGBDBM698752(US20240317732, Compound XL30)
Affinity DataKd:  1.24E+4nMAssay Description:ITC experiments were performed at 25° C. on a MicroCal iTC200 system (Malvern, PA, USA). hRpn13 Pru, XL5, XL5 derivative, or RA190 were prepared in b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/28/2025
Entry Details
Go to US Patent