Compile Data Set for Download or QSAR
Report error Found 99 Enz. Inhib. hit(s) with all data for entry = 12206
TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686544(US20240246935, Example 124 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  2nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686471(3-(5-(((1S,2S)-2-(3-(4- fluorophenyl)azetidin-1- y...)
Affinity DataEC50:  4nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686547(US20240246935, Example 130 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  4nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686547(US20240246935, Example 130 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  4nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686546(US20240246935, Example 126 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  5nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686494(US20240246935, Example 73 | 3-(5-(((1S,2S)-2-(3-(4...)
Affinity DataEC50:  5nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686468(US20240246935, Example 48 | US20240246935, Example...)
Affinity DataEC50:  5nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686545(US20240246935, Example 125 | (R)-3-(1-oxo-5-(((1S,...)
Affinity DataEC50:  6nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686478(US20240246935, Example 57 | 3-(5-(((1S,2S)-2-(3-(2...)
Affinity DataEC50:  6nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686541(US20240246935, Example 121 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  6nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686532(US20240246935, Example 111 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  6nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686493(US20240246935, Example 72 | 3-(1-oxo-5-(((1S,2S)-2...)
Affinity DataEC50:  7nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686459(US20240246935, Example 99 | US20240246935, Example...)
Affinity DataEC50:  8nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686539(US20240246935, Example 119 | Rac-4-(1-((trans)-2-(...)
Affinity DataEC50:  8nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686501(US20240246935, Example 80 | 3-(5-(((1S,2S)-2-(3-(3...)
Affinity DataEC50:  8nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686502(US20240246935, Example 81 | 3-(5-(((1S,2S)-2-(3-(4...)
Affinity DataEC50:  9nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686480(US20240246935, Example 59 | 3-(1-oxo-5-(((1R,2S)-2...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686471(3-(5-(((1S,2S)-2-(3-(4- fluorophenyl)azetidin-1- y...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686540(US20240246935, Example 120 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686461(US20240246935, Example 40 | 5-chloro-2-(1-((1S,2R)...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686552(US20240246935, Example 132 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686551(US20240246935, Example 131 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686473(US20240246935, Example 53 | 3-(6-fluoro-1-oxo-5-((...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686470(US20240246935, Example 49 | 3-chloro-4-(1-((1S,2R)...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686485(US20240246935, Example 64 | 3-(5-(((1S,2S)-2-(3-(2...)
Affinity DataEC50:  11nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686496(US20240246935, Example 75 | Rac-3-chloro-4-(1-((ci...)
Affinity DataEC50:  12nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686535(US20240246935, Example 115 | Rac-4-(1-((cis)-2-((2...)
Affinity DataEC50:  12nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686554(US20240246935, Example 134 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  12nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686500(US20240246935, Example 79 | 3-(1-oxo-5-(((1S,2S)-2...)
Affinity DataEC50:  12nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686534(US20240246935, Example 113 | 3-(1-((1S,2S)-2-((2-(...)
Affinity DataEC50:  13nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686482(US20240246935, Example 61 | Rac-3-(1-oxo-5-(((cis)...)
Affinity DataEC50:  14nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686553(US20240246935, Example 133 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  14nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686505(US20240246935, Example 84 | Rac-5-chloro-2-(1-((ci...)
Affinity DataEC50:  14nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686481(Rac-3-(1-oxo-5-(((trans)-2-(3-(4- (trifluoromethox...)
Affinity DataEC50:  15nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686524(US20240246935, Example 103 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  15nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686484(US20240246935, Example 63 | Rac-3-(1-oxo-5-(((cis)...)
Affinity DataEC50:  15nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686456(US20240246935, Example 35 | 3-(1-oxo-5-(((1S,2S)-2...)
Affinity DataEC50:  17nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686488(US20240246935, Example 67 | 3-(1-oxo-5-((2-(3-(3- ...)
Affinity DataEC50:  17nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686549(US20240246935, Example 129 | 3-(1-oxo-5-(((1S,2S)-...)
Affinity DataEC50:  17nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686525(US20240246935, Example 104 | 3-(5-(((1S,2S)-2-(3-(...)
Affinity DataEC50:  18nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686471(3-(5-(((1S,2S)-2-(3-(4- fluorophenyl)azetidin-1- y...)
Affinity DataEC50:  18nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686548(US20240246935, Example 128 | 3-(1-oxo-5-(((1S,2R)-...)
Affinity DataEC50:  18nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686531(US20240246935, Example 110 | 4-(1-(2-((2-(2,6-diox...)
Affinity DataEC50:  19nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686468(US20240246935, Example 48 | US20240246935, Example...)
Affinity DataEC50:  20nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686542(US20240246935, Example 122 | Rac-4-(1-((cis)-2-((2...)
Affinity DataEC50:  20nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686465(US20240246935, Example 45 | US20240246935, Example...)
Affinity DataEC50:  22nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686497(US20240246935, Example 76 | Rac-3-(1-((cis)-2-((2-...)
Affinity DataEC50:  22nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686467(2-(1-((1S,2R)-2-((2-(2,6- dioxopiperidin-3-yl)-1- ...)
Affinity DataEC50:  22nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686467(2-(1-((1S,2R)-2-((2-(2,6- dioxopiperidin-3-yl)-1- ...)
Affinity DataEC50:  24nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

TargetProtein cereblon(Human)
Plexium, Inc.

US Patent
LigandPNGBDBM686536(US20240246935, Example 116 | Rac-4-(1-((trans)-2-(...)
Affinity DataEC50:  24nMAssay Description:Cereblon target engagement was monitored by Bioluminescence Resonance Energy Transfer (BRET) in transfected HEK-293T cells using the NanoBRET TE Intr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/7/2024
Entry Details
Go to US Patent

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