Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 12043
TargetSynaptic vesicular amine transporter(Rat)
Columbia University

US Patent
LigandPNGBDBM674463(US20240150372, Compound (16R)-Oxa-noribogaine)
Affinity DataIC50: 140nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetSodium-dependent serotonin transporter(Human)
Columbia University

US Patent
LigandPNGBDBM674463(US20240150372, Compound (16R)-Oxa-noribogaine)
Affinity DataIC50: 450nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetSynaptic vesicular amine transporter(Rat)
Columbia University

US Patent
LigandPNGBDBM674461(US20240150372, Compound Oxa-noribogaine)
Affinity DataIC50: 670nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetSodium-dependent serotonin transporter(Human)
Columbia University

US Patent
LigandPNGBDBM674461(US20240150372, Compound Oxa-noribogaine)
Affinity DataIC50: 900nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetSynaptic vesicular amine transporter(Rat)
Columbia University

US Patent
LigandPNGBDBM674462(US20240150372, Compound (16S)-Oxa-noribogaine)
Affinity DataIC50: 2.80E+3nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetSodium-dependent serotonin transporter(Human)
Columbia University

US Patent
LigandPNGBDBM674462(US20240150372, Compound (16S)-Oxa-noribogaine)
Affinity DataIC50: 2.90E+3nMAssay Description:hSERT and rVMAT2 fluorometric screening assays. For both hSERT and rVMAT2 screening experiments, respective singly transfected cells were seeded at a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent