Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 12036
TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM633575((S) N ((S)-1-cyano-2-(2-fluoro-4-(3-methyl-2-oxo-2...)
Affinity DataIC50: 0.640nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674394(US20240150335, Compound 22)
Affinity DataIC50: 0.760nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM633575((S) N ((S)-1-cyano-2-(2-fluoro-4-(3-methyl-2-oxo-2...)
Affinity DataIC50: 0.840nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674395(US20240150335, Compound 24)
Affinity DataIC50: 1nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674390(US20240150335, Compound 18)
Affinity DataIC50: 1.23nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674377(US20240150335, Compound 4)
Affinity DataIC50: 1.32nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674384(US20240150335, Compound 12)
Affinity DataIC50: 1.81nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674384(US20240150335, Compound 12)
Affinity DataIC50: 2.38nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674381(US20240150335, Compound 8)
Affinity DataIC50: 2.40nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674380(US20240150335, Compound 7)
Affinity DataIC50: 2.49nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674380(US20240150335, Compound 7)
Affinity DataIC50: 2.52nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674386(US20240150335, Compound 14)
Affinity DataIC50: 2.79nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674395(US20240150335, Compound 24)
Affinity DataIC50: 3.12nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674381(US20240150335, Compound 8)
Affinity DataIC50: 3.57nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674387(US20240150335, Compound 15)
Affinity DataIC50: 3.65nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674383(US20240150335, Compound 10)
Affinity DataIC50: 4.39nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674391(US20240150335, Compound 19)
Affinity DataIC50: 4.55nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674390(US20240150335, Compound 18)
Affinity DataIC50: 5.43nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674385(US20240150335, Compound 13)
Affinity DataIC50: 6.33nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674383(US20240150335, Compound 10)
Affinity DataIC50: 8.53nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674391(US20240150335, Compound 19)
Affinity DataIC50: 8.70nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674376(US20240150335, Compound 2)
Affinity DataIC50: 8.95nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674388(US20240150335, Compound 16)
Affinity DataIC50: 9.18nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674393(US20240150335, Compound 21)
Affinity DataIC50: 9.27nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674378(US20240150335, Compound 5)
Affinity DataIC50: 9.32nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674392(US20240150335, Compound 20)
Affinity DataIC50: 9.58nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674377(US20240150335, Compound 4)
Affinity DataIC50: 10.8nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674392(US20240150335, Compound 20)
Affinity DataIC50: 11.5nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674382(US20240150335, Compound 9)
Affinity DataIC50: 14nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674393(US20240150335, Compound 21)
Affinity DataIC50: 17.3nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674385(US20240150335, Compound 13)
Affinity DataIC50: 20.4nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674389(US20240150335, Compound 17)
Affinity DataIC50: 22.5nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674376(US20240150335, Compound 2)
Affinity DataIC50: 26.8nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674386(US20240150335, Compound 14)
Affinity DataIC50: 28.1nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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TargetDipeptidyl peptidase 1(Human)
Medshine Discovery

US Patent
LigandPNGBDBM674378(US20240150335, Compound 5)
Affinity DataIC50: 28.3nMAssay Description:Experimental Methods:1× activation buffer: 5 mM DTT 0.01% (V/V) Triton X-100 (preparation for current use);1× assay buffer: 50 mM NaCl 5 mM DTT 0.01%...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
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