Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 12033
TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673766(US20240150300, Compound I-2)
Affinity DataIC50: 23.3nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673782(US20240150300, Compound I-12)
Affinity DataIC50: 31.3nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673772(US20240150300, Compound I-4)
Affinity DataIC50: 35.2nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673768(US20240150300, Compound HYH-072 (racemate of I-2))
Affinity DataIC50: 38.3nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673781(US20240150300, Compound I-11)
Affinity DataIC50: 42.4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673783(US20240150300, Compound I-13)
Affinity DataIC50: 44.8nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673779(US20240150300, Compound I-10)
Affinity DataIC50: 50.5nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673770(US20240150300, Compound I-3)
Affinity DataIC50: 52.4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673763(US20240150300, Compound I-1)
Affinity DataIC50: 57.6nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673775(US20240150300, Compound I-6)
Affinity DataIC50: 60.5nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673769(US20240150300, Compound I-2(R configuration))
Affinity DataIC50: 72.1nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673764(US20240150300, Compound HYH-073 (racemate of I-1))
Affinity DataIC50: 80.5nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673771(US20240150300, Compound I-3(racemic))
Affinity DataIC50: 81.9nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673763(US20240150300, Compound I-1)
Affinity DataIC50: 90nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673766(US20240150300, Compound I-2)
Affinity DataIC50: 90nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673776(US20240150300, Compound I-7)
Affinity DataIC50: 99.5nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673773(US20240150300, Compound I-4(racemic))
Affinity DataIC50: 107nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673778(US20240150300, Compound I-9)
Affinity DataIC50: 122nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673774(US20240150300, Compound I-5)
Affinity DataIC50: 124nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673777(US20240150300, Compound I-8)
Affinity DataIC50: 126nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM50242817(CHEMBL4087968 | US20240150300, Compound Chidamide)
Affinity DataIC50: 132nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673780(US20240150300, Compound I-10(R configuration))
Affinity DataIC50: 155nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 255nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673769(US20240150300, Compound I-2(R configuration))
Affinity DataIC50: 300nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673765(US20240150300, Compound I-1 (R configuration))
Affinity DataIC50: 320nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 1(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673765(US20240150300, Compound I-1 (R configuration))
Affinity DataIC50: 375nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673766(US20240150300, Compound I-2)
Affinity DataIC50: 390nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673763(US20240150300, Compound I-1)
Affinity DataIC50: 420nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673765(US20240150300, Compound I-1 (R configuration))
Affinity DataIC50: 720nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 2(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 750nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673769(US20240150300, Compound I-2(R configuration))
Affinity DataIC50: 840nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 3(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 1.58E+3nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673782(US20240150300, Compound I-12)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673763(US20240150300, Compound I-1)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673783(US20240150300, Compound I-13)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM19410(benzamide-type inhibitor, 3 | CHEMBL27759 | pyridi...)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM50242817(CHEMBL4087968 | US20240150300, Compound Chidamide)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673780(US20240150300, Compound I-10(R configuration))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673766(US20240150300, Compound I-2)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673768(US20240150300, Compound HYH-072 (racemate of I-2))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673769(US20240150300, Compound I-2(R configuration))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673770(US20240150300, Compound I-3)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673765(US20240150300, Compound I-1 (R configuration))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673764(US20240150300, Compound HYH-073 (racemate of I-1))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673771(US20240150300, Compound I-3(racemic))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673772(US20240150300, Compound I-4)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673781(US20240150300, Compound I-11)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673773(US20240150300, Compound I-4(racemic))
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673774(US20240150300, Compound I-5)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

TargetHistone deacetylase 6(Human)
Shanghai Institute of Materia Medica

US Patent
LigandPNGBDBM673775(US20240150300, Compound I-6)
Affinity DataIC50: 1.00E+4nMAssay Description:Human recombinant HDAC family proteins with His and GST tags were expressed using insect baculovirus expression system, and a biologically active HDA...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/9/2024
Entry Details
Go to US Patent

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