Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 4657
TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM191600(US9714230, 89 | 2-(5-((4-chloro-2-methylbenzyl)oxy...)
Affinity DataIC50: 2nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264012(2-[5-[(4-chloro-2- methoxyphenyl)methoxy]pyrazol- ...)
Affinity DataIC50: 3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670395(US20240139197, Compound 37)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264030(2-[5-[(4-chloro-2- ethoxyphenyl)methoxy]pyrazol-1-...)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670388(US20240139197, Compound 21)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264001(2-{5-[(4-chloro-2- fluorobenzyl)oxy]-1H-pyrazol-1-...)
Affinity DataIC50: 4nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532176(CHEMBL4542928 | US20240139197, Compound 13)
Affinity DataIC50: 4.37nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264012(2-[5-[(4-chloro-2- methoxyphenyl)methoxy]pyrazol- ...)
Affinity DataIC50: 12nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM191600(US9714230, 89 | 2-(5-((4-chloro-2-methylbenzyl)oxy...)
Affinity DataIC50: 13nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670388(US20240139197, Compound 21)
Affinity DataIC50: 14nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264001(2-{5-[(4-chloro-2- fluorobenzyl)oxy]-1H-pyrazol-1-...)
Affinity DataIC50: 18nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264030(2-[5-[(4-chloro-2- ethoxyphenyl)methoxy]pyrazol-1-...)
Affinity DataIC50: 18nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532173(CHEMBL4536443 | US20240139197, Compound 10)
Affinity DataIC50: 22.7nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264022(2-[5-[[4-chloro-2- (cyclopropylmethoxy(phenyl] met...)
Affinity DataIC50: 25nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670395(US20240139197, Compound 37)
Affinity DataIC50: 32nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5B(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264022(2-[5-[[4-chloro-2- (cyclopropylmethoxy(phenyl] met...)
Affinity DataIC50: 36nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264012(2-[5-[(4-chloro-2- methoxyphenyl)methoxy]pyrazol- ...)
Affinity DataIC50: 38nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM191600(US9714230, 89 | 2-(5-((4-chloro-2-methylbenzyl)oxy...)
Affinity DataIC50: 41nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670388(US20240139197, Compound 21)
Affinity DataIC50: 54nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532175(CHEMBL4436444 | US20240139197, Compound 11)
Affinity DataIC50: 65.3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM670395(US20240139197, Compound 37)
Affinity DataIC50: 74nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264030(2-[5-[(4-chloro-2- ethoxyphenyl)methoxy]pyrazol-1-...)
Affinity DataIC50: 78nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532943(CHEMBL4449759 | US20240139197, Compound 7)
Affinity DataIC50: 170nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532177(CHEMBL4556977 | US20240139197, Compound 12)
Affinity DataIC50: 179nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 4C(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM264022(2-[5-[[4-chloro-2- (cyclopropylmethoxy(phenyl] met...)
Affinity DataIC50: 280nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent

TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM195608(CPI-455 | US20240139197, Compound 3)
Affinity DataIC50: 506nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent
PDB3D3D Structure (crystal)
TargetLysine-specific demethylase 5A(Human)
The Wistar Institute of Anatomy and Biology

US Patent
LigandPNGBDBM50532943(CHEMBL4449759 | US20240139197, Compound 7)
Affinity DataIC50: 2.70E+3nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/2/2024
Entry Details
Go to US Patent