Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 12010
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889(US20240132517, Example 1 | (S, 13E, 14E)-2-ethyl-4...)
Affinity DataIC50: 0.420nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889(US20240132517, Example 1 | (S, 13E, 14E)-2-ethyl-4...)
Affinity DataIC50: 0.930nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888(US20240132517, Example TPX-0022 | Example 5 of WO...)
Affinity DataIC50: 1.80nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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PDB3D3D Structure (crystal)
TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890(US20240132517, Example 2 | (S, 13E, 14E)-12-amino-...)
Affinity DataIC50: 1.80nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890(US20240132517, Example 2 | (S, 13E, 14E)-12-amino-...)
Affinity DataIC50: 2.20nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888(US20240132517, Example TPX-0022 | Example 5 of WO...)
Affinity DataIC50: 7.5nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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PDB3D3D Structure (crystal)
TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669888(US20240132517, Example TPX-0022 | Example 5 of WO...)
Affinity DataIC50: 10nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669889(US20240132517, Example 1 | (S, 13E, 14E)-2-ethyl-4...)
Affinity DataIC50: 15nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669890(US20240132517, Example 2 | (S, 13E, 14E)-12-amino-...)
Affinity DataIC50: 30nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetHepatocyte growth factor receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42 | US1212925...)
Affinity DataIC50: 85nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetProto-oncogene tyrosine-protein kinase Src(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42 | US1212925...)
Affinity DataIC50: 289nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
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TargetMacrophage colony-stimulating factor 1 receptor(Human)
Goharmony Therapeutics (Shenzhen) Co.

US Patent
LigandPNGBDBM669891(US20240132517, Comparative Compound 42 | US1212925...)
Affinity DataIC50: 1.00E+4nMAssay Description:The operation method is briefly described as follows:The powders of the compound were dissolved in 100% DMSO to make a 10 mM stock solution. The init...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/16/2024
Entry Details
Go to US Patent