Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 11740
TargetTyrosine-protein kinase BTK [C481S](Human)
Haisco Pharmaceuticals

US Patent
LigandPNGBDBM588276(5-[3-[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,...)
Affinity DataIC50: 6.30nMAssay Description:Conclusion: compound 1 had a significant inhibitory effect on BTK wt/C481S kinase.More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetTyrosine-protein kinase BTK(Human)
Haisco Pharmaceuticals

US Patent
LigandPNGBDBM588276(5-[3-[3-[4-[4-amino-3-(4-phenoxyphenyl)pyrazolo[3,...)
Affinity DataIC50: 8nMAssay Description:Conclusion: compound 1 had a significant inhibitory effect on BTK wt/C481S kinase.More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent