Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 11738
TargetTyrosine-protein kinase BTK [C481S](Human)
Medshine Discovery

US Patent
LigandPNGBDBM643175(US20240002377, Compound 4)
Affinity DataIC50: 7.40nMAssay Description:1. The substrate was prepared in freshly prepared reaction buffer;2. The required cofactor was added to the above-mentioned substrate solution;3. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK [C481S](Human)
Medshine Discovery

US Patent
LigandPNGBDBM643176(US20240002377, Compound 5)
Affinity DataIC50: 8.90nMAssay Description:1. The substrate was prepared in freshly prepared reaction buffer;2. The required cofactor was added to the above-mentioned substrate solution;3. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK [C481S](Human)
Medshine Discovery

US Patent
LigandPNGBDBM643173(US20240002377, Compound 2)
Affinity DataIC50: 11.7nMAssay Description:1. The substrate was prepared in freshly prepared reaction buffer;2. The required cofactor was added to the above-mentioned substrate solution;3. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK [C481S](Human)
Medshine Discovery

US Patent
LigandPNGBDBM643172(US20240002377, Compound 1)
Affinity DataIC50: 58.9nMAssay Description:1. The substrate was prepared in freshly prepared reaction buffer;2. The required cofactor was added to the above-mentioned substrate solution;3. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent

TargetTyrosine-protein kinase BTK [C481S](Human)
Medshine Discovery

US Patent
LigandPNGBDBM643174(US20240002377, Compound 3)
Affinity DataIC50: 74.2nMAssay Description:1. The substrate was prepared in freshly prepared reaction buffer;2. The required cofactor was added to the above-mentioned substrate solution;3. The...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent