Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 11736
TargetFibroblast growth factor receptor 2(Human)
Beta Pharma

US Patent
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 0.800nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Beta Pharma

US Patent
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.10nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 2(Human)
Beta Pharma

US Patent
LigandPNGBDBM643160(US20240002365, Example 1 | N1-(3,5-Dimethoxyphenyl...)
Affinity DataIC50: 4.30nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Beta Pharma

US Patent
LigandPNGBDBM643160(US20240002365, Example 1 | N1-(3,5-Dimethoxyphenyl...)
Affinity DataIC50: 7.30nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Beta Pharma

US Patent
LigandPNGBDBM643160(US20240002365, Example 1 | N1-(3,5-Dimethoxyphenyl...)
Affinity DataIC50: 7.60nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Beta Pharma

US Patent
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 8.90nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Beta Pharma

US Patent
LigandPNGBDBM643160(US20240002365, Example 1 | N1-(3,5-Dimethoxyphenyl...)
Affinity DataIC50: 9.5nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Beta Pharma

US Patent
LigandPNGBDBM643160(US20240002365, Example 1 | N1-(3,5-Dimethoxyphenyl...)
Affinity DataIC50: 11nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
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Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 1(Human)
Beta Pharma

US Patent
LigandPNGBDBM50592470(CHEMBL5189795 | US20240002365, Compound CTx-029488...)
Affinity DataIC50: 35nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
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TargetFibroblast growth factor receptor 4(Human)
Beta Pharma

US Patent
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 41nMAssay Description:The reaction procedure was conducted as follows:1) Prepare substrate in freshly prepared Reaction Buffer.2) MnCl2 (2 mM) was added as a co-factor lis...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
Go to US Patent