Compile Data Set for Download or QSAR
Report error Found 27 Enz. Inhib. hit(s) with all data for entry = 11700
TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640922((S)-4-(8-(3-aminopiperidin-1-yl)-3-(1-(2-ethyl-2-h...)
Affinity DataIC50: 0.700nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640917((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-(2-...)
Affinity DataIC50: 0.710nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640907((R)-4-(8-(3-aminopiperidin-1-yl)-3-(4-methyll-3,4-...)
Affinity DataIC50: 0.880nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640909((R)-4-(8-(3-aminopiperidin-1-yl)-3-(1-(2-hydroxy-2...)
Affinity DataIC50: 0.970nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640925((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-met...)
Affinity DataIC50: 1nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640923(4-(8-((1S,2S,4R)-2-amino-7-azabicyclo[2.2.1]heptan...)
Affinity DataIC50: 1nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640902((R)4-(7-(3-aminopiperidin-1-yl)-3-(3-fluoro-4-meth...)
Affinity DataIC50: 1nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640900((R)-4-(8-(3-aminopiperidin-1-yl)-3-(3-fluoro-4-met...)
Affinity DataIC50: 1.30nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640910((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-(2-...)
Affinity DataIC50: 1.60nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640906((R)-4-(8-(3-aminopiperidin-1-yl)-3-(1-methyll-1H-i...)
Affinity DataIC50: 1.70nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640903((R)-4-(8-(3-aminopiperidin-1-yl)-3-(1-methyll-1H-i...)
Affinity DataIC50: 2.30nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640919((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-2-(2-...)
Affinity DataIC50: 2.30nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640920((R)-4-(8-(3-aminopiperidin-1-yl)-3-(2-fluoro-4-(2-...)
Affinity DataIC50: 2.5nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640901(4-(7-(4-aminopiperidin-1-yl)-3-(3-fluoro-4-methoxy...)
Affinity DataIC50: 2.60nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640918((R)-4-(8-(3-aminopiperidin-1-yl)-3-(1-(2-hydroxy-2...)
Affinity DataIC50: 2.60nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640916((R)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-(2-...)
Affinity DataIC50: 2.90nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640921((S)-4-(8-(3-aminopiperidin-1-yl)-3-(6-fluoro-1-(2-...)
Affinity DataIC50: 4.40nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640924(((1R,3r,5S)-8-(2-(4-cyano-3-fluorophenyl)-3-(6-flu...)
Affinity DataIC50: 5.5nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640915((R)-4-(8-(3-aminopiperidin-1-yl)-3-(2-methyll-2H-i...)
Affinity DataIC50: 6.30nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640899(4-(8-(4-aminopiperidin-1-yl)-3-(3-fluoro-4-methoxy...)
Affinity DataIC50: 7.40nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640908((R)-4-(8-(3-aminopiperidin-1-yl)-3-(1-(2,2,2-trifl...)
Affinity DataIC50: 7.5nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640913(trans-4-(8-(((1R,3R)-3-aminocyclopentyl)amino)-3-(...)
Affinity DataIC50: 11nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640905(2-fluoro-4-(3-(3-fluoro-4-methoxyphenyl)-8-(piperi...)
Affinity DataIC50: 12nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640914(2-fluoro-4-(3-(3-fluoro-4-methoxyphenyl)-8-(pyrrol...)
Affinity DataIC50: 15nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
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Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640912(cis-4-(8-(((1R,3S)-3-aminocyclopentyl)amino)-3-(3-...)
Affinity DataIC50: 37nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640904(2-fluoro-4-(3-(3-fluoro-4-methoxyphenyl)-8-((pyrro...)
Affinity DataIC50: 45nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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TargetLysine-specific histone demethylase 1A(Human)
Tencent Technology (Shenzhen)

US Patent
LigandPNGBDBM640911(2-fluoro-4-(3-(3-fluoro-4-methoxyphenyl)-8-((pyrro...)
Affinity DataIC50: 56nMAssay Description:Experimental steps and a method: In this experiment, the in vitro inhibitory activity of the compounds of the present disclosure against LSD1 on an e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/3/2024
Entry Details
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