Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 11655
TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636827(US20230382869, Compound Table1.1 | US20230382869, ...)
Affinity DataEC50:  8.28nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636828(US20230382869, Compound Table1.2 | US20230382869, ...)
Affinity DataEC50:  7.96nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636829(US20230382869, Compound Table1.3 | 2-(2-chloro-6-f...)
Affinity DataEC50:  13.2nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636830(US20230382869, Compound Table1.4 | 2-(2,6-dichloro...)
Affinity DataEC50:  5.19nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636831(US20230382869, Compound Table1.5 | 2-(2-chloro-6-f...)
Affinity DataEC50:  10.2nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636827(US20230382869, Compound Table1.1 | US20230382869, ...)
Affinity DataEC50:  12.1nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636833(US20230382869, Compound Table1.7 | US20230382869, ...)
Affinity DataEC50:  11.2nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636833(US20230382869, Compound Table1.7 | US20230382869, ...)
Affinity DataEC50:  86.7nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636828(US20230382869, Compound Table1.2 | US20230382869, ...)
Affinity DataEC50:  12.7nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636836(US20230382869, Compound Table1.10 | 2-(2-chloro-6-...)
Affinity DataEC50:  33.6nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
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TargetD(1A) dopamine receptor(Human)
Eli Lilly

US Patent
LigandPNGBDBM636830(US20230382869, Compound Table1.4 | 2-(2,6-dichloro...)
Affinity DataEC50:  12.3nMAssay Description:Test compound is serially diluted (1:2) with DMSO into assay plates (ProxiPlate-384 Plus, PerkinElmer) using acoustic dispensing (Labcyte) to provide...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/19/2024
Entry Details
Go to US Patent