Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 11583
TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628884(US20230339896, Example 2)
Affinity DataIC50: 0.200nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
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TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628887(US20230339896, Example 5)
Affinity DataIC50: 0.200nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
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TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628883(US20230339896, Example 1)
Affinity DataIC50: 0.5nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628891(US20230339896, Example 10)
Affinity DataIC50: 0.5nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628886(US20230339896, Example 4)
Affinity DataIC50: 0.700nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
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TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628888(US20230339896, Example 7)
Affinity DataIC50: 1nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628890(US20230339896, Example 9)
Affinity DataIC50: 1.10nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628889(US20230339896, Example 8)
Affinity DataIC50: 1.5nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase kinase kinase kinase 1(Human)
Qilu Regor Therapeutics

US Patent
LigandPNGBDBM628885(US20230339896, Example 3)
Affinity DataIC50: 24nMAssay Description:The ADP-GLO Kinase Assay (Promega Corp., Madison, WI) measures ADP formed from a kinase reaction. According to the manufacture, the ADP formed in a k...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/10/2023
Entry Details
Go to US Patent