Compile Data Set for Download or QSAR
Report error Found 2 Enz. Inhib. hit(s) with all data for entry = 11509
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Human)
Guangzhou Baiyunshan Pharmaceutical Holdings Co., Ltd. Baiyunshan Pharmaceutical General Factory

US Patent
LigandPNGBDBM621734(US20230312504, Compound 1)
Affinity DataIC50: 0.5nMAssay Description:The inhibitory activity of the test compounds against human wild-type and V804M mutant RET kinase was evaluated by measuring IC50 values in a 33P-lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
Go to US Patent

TargetProto-oncogene tyrosine-protein kinase receptor Ret [V804M](Human)
Guangzhou Baiyunshan Pharmaceutical Holdings Co., Ltd. Baiyunshan Pharmaceutical General Factory

US Patent
LigandPNGBDBM621734(US20230312504, Compound 1)
Affinity DataIC50: 0.900nMAssay Description:The inhibitory activity of the test compounds against human wild-type and V804M mutant RET kinase was evaluated by measuring IC50 values in a 33P-lab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/13/2023
Entry Details
Go to US Patent