Compile Data Set for Download or QSAR
Report error Found 1 Enz. Inhib. hit(s) with all data for entry = 5843
TargetSerine/threonine-protein kinase ATR(Human)
Vertex Pharmaceuticals

US Patent
LigandPNGBDBM97372(US20130089624, 1)
Affinity DataKi:  0.503nM ΔG°:  -53.1kJ/mole IC50: 200nMpH: 7.5 T: 2°CAssay Description:Assays were carried out in a mixture of 50 mM Tris/HCl (pH 7.5), 10 mM MgCl2 and 1 mM DTT. Final substrate concentrations were 10 μM [γ-33P]...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2013
Entry Details
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