Compile Data Set for Download or QSAR
Report error Found 53 Enz. Inhib. hit(s) with all data for entry = 13301
Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564453(CHEMBL4794096 | US12435059, Compound 17)
Affinity DataIC50: 16.2nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564457(CHEMBL4800500 | US12435059, Compound 10)
Affinity DataIC50: 20.5nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564458(CHEMBL4788376 | US12435059, Compound 15)
Affinity DataIC50: 32.4nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564448(CHEMBL4788980 | US12435059, Compound 8)
Affinity DataIC50: 38.6nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564449(CHEMBL4779166 | US12435059, Compound 20)
Affinity DataIC50: 49.4nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM4817(N-[2-(dimethylamino)ethyl]-5-{[(3Z)-5-fluoro-2-oxo...)
Affinity DataIC50: 50.4nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564459(CHEMBL4781578 | US12435059, Compound 16)
Affinity DataIC50: 60.7nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564446(CHEMBL3542344 | US12435059, Compound 6)
Affinity DataIC50: 61.4nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 61.7nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564450(CHEMBL4786972 | US12435059, Compound 21)
Affinity DataIC50: 65.1nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564447(CHEMBL4799580 | US12435059, Compound 7)
Affinity DataIC50: 74.8nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564451(CHEMBL4782796 | US12435059, Compound 22)
Affinity DataIC50: 82.5nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564454(CHEMBL4792246 | US12435059, Compound 18)
Affinity DataIC50: 83.6nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM4813(N-[2-(diethylamino)ethyl]-2,4-dimethyl-5-{[(3Z)-2-...)
Affinity DataIC50: 88.5nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564453(CHEMBL4794096 | US12435059, Compound 17)
Affinity DataIC50: 93nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564455(CHEMBL4781062 | US12435059, Compound 9)
Affinity DataIC50: 96.6nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564462(CHEMBL4796639 | US12435059, Compound 13)
Affinity DataIC50: 101nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564459(CHEMBL4781578 | US12435059, Compound 16)
Affinity DataIC50: 107nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564461(CHEMBL4795330 | US12435059, Compound 14)
Affinity DataIC50: 108nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564456(CHEMBL4799631 | US12435059, Compound 11)
Affinity DataIC50: 111nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM4817(N-[2-(dimethylamino)ethyl]-5-{[(3Z)-5-fluoro-2-oxo...)
Affinity DataIC50: 136nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564462(CHEMBL4796639 | US12435059, Compound 13)
Affinity DataIC50: 139nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564445(CHEMBL3542333 | US12435059, Compound 4)
Affinity DataIC50: 141nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564448(CHEMBL4788980 | US12435059, Compound 8)
Affinity DataIC50: 152nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564460(CHEMBL4779730 | US12435059, Compound 12)
Affinity DataIC50: 154nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 158nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564458(CHEMBL4788376 | US12435059, Compound 15)
Affinity DataIC50: 164nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564457(CHEMBL4800500 | US12435059, Compound 10)
Affinity DataIC50: 173nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564446(CHEMBL3542344 | US12435059, Compound 6)
Affinity DataIC50: 180nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564461(CHEMBL4795330 | US12435059, Compound 14)
Affinity DataIC50: 184nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564449(CHEMBL4779166 | US12435059, Compound 20)
Affinity DataIC50: 189nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564454(CHEMBL4792246 | US12435059, Compound 18)
Affinity DataIC50: 205nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564450(CHEMBL4786972 | US12435059, Compound 21)
Affinity DataIC50: 206nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564451(CHEMBL4782796 | US12435059, Compound 22)
Affinity DataIC50: 208nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564450(CHEMBL4786972 | US12435059, Compound 21)
Affinity DataIC50: 217nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564447(CHEMBL4799580 | US12435059, Compound 7)
Affinity DataIC50: 221nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564449(CHEMBL4779166 | US12435059, Compound 20)
Affinity DataIC50: 240nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM4813(N-[2-(diethylamino)ethyl]-2,4-dimethyl-5-{[(3Z)-2-...)
Affinity DataIC50: 246nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564455(CHEMBL4781062 | US12435059, Compound 9)
Affinity DataIC50: 296nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564452(CHEMBL4785831 | US12435059, Compound 24)
Affinity DataIC50: 348nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564453(CHEMBL4794096 | US12435059, Compound 17)
Affinity DataIC50: 391nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564445(CHEMBL3542333 | US12435059, Compound 4)
Affinity DataIC50: 393nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564456(CHEMBL4799631 | US12435059, Compound 11)
Affinity DataIC50: 418nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM4814(SUNITINIB MALATE | CHEMBL535 | N-[2-(diethylamino)...)
Affinity DataIC50: 461nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564448(CHEMBL4788980 | US12435059, Compound 8)
Affinity DataIC50: 480nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM4817(N-[2-(dimethylamino)ethyl]-5-{[(3Z)-5-fluoro-2-oxo...)
Affinity DataIC50: 493nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564446(CHEMBL3542344 | US12435059, Compound 6)
Affinity DataIC50: 505nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564457(CHEMBL4800500 | US12435059, Compound 10)
Affinity DataIC50: 848nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

TargetVascular endothelial growth factor receptor 2(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564458(CHEMBL4788376 | US12435059, Compound 15)
Affinity DataIC50: 1.33E+3nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

Target5'-AMP-activated protein kinase catalytic subunit alpha-1(Human)
University Of Colorado

US Patent
LigandPNGBDBM50564460(CHEMBL4779730 | US12435059, Compound 12)
Affinity DataIC50: 2.10E+3nMAssay Description:LANCE® Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assays (PerkinElmer) were performed in 384-well OptiPlates (Corning) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/21/2026
Entry Details
US Patent

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