Compile Data Set for Download or QSAR
Report error Found 11 Enz. Inhib. hit(s) with all data for entry = 13256
TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771610(US12415819, Compound 58)
Affinity DataIC50: 0.0110nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771604(US12415819, Compound 52-B(OH)2)
Affinity DataIC50: 0.0150nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771602(US12415819, Compound 51-B(OH)2)
Affinity DataIC50: 0.0300nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM50120437(CHEMBL3617973 | US12415819, Compound 54)
Affinity DataIC50: 0.0310nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771607(POL6014 | US12415819, Compound 55)
Affinity DataIC50: 0.0930nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM50608626(CHEMBL5280380 | US12415819, Compound 50-B(OH)2)
Affinity DataIC50: 0.270nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771609(US12415819, Compound 57)
Affinity DataIC50: 0.990nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM771608(US12415819, Compound 56)
Affinity DataIC50: 1.34nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM50120430(CHEMBL3617964 | US12415819, Compound 53)
Affinity DataIC50: 2.62nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM50061024((2-Methyl-1-{(S)-oxo-[(S)-2-((S)-3,3,3-trifluoro-1...)
Affinity DataIC50: 135nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent

TargetNeutrophil elastase(Human)
The Scripps Research Institute

US Patent
LigandPNGBDBM50031201((S)-1-{(S)-2-[4-(4-Chloro-benzenesulfonylaminocarb...)
Affinity DataIC50: 290nMAssay Description:Serially diluted compounds in DMSO were dispensed into a 384-well black opaque plate by Echo dispenser. 0.1 μg/mL human neutrophil elastase (EPC, Cat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/29/2025
Entry Details
US Patent