Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 12648
TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717677(US12215095, Compound ZH2-102)
Affinity DataIC50: 1.70nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717677(US12215095, Compound ZH2-102)
Affinity DataIC50: 1.70nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717678(US12215095, Compound ZH2-130)
Affinity DataIC50: 1.93nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717678(US12215095, Compound ZH2-130)
Affinity DataIC50: 1.95nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717686(US12215095, Compound ZH3-98)
Affinity DataIC50: 2.54nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717686(US12215095, Compound ZH3-98)
Affinity DataIC50: 2.57nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717683(US12215095, Compound ZH3-74)
Affinity DataIC50: 2.95nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717683(US12215095, Compound ZH3-74)
Affinity DataIC50: 2.97nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717688(US12215095, Compound ZH2-122)
Affinity DataIC50: 5.07nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717681(US12215095, Compound ZH2-86)
Affinity DataIC50: 7.08nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717681(US12215095, Compound ZH2-86)
Affinity DataIC50: 7.16nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717682(US12215095, Compound ZH2-98)
Affinity DataIC50: 12.3nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717682(US12215095, Compound ZH2-98)
Affinity DataIC50: 12.6nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717685(US12215095, Compound ZH3-94)
Affinity DataIC50: 34.4nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717685(US12215095, Compound ZH3-94)
Affinity DataIC50: 34.7nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717679(US12215095, Compound ZH2-62)
Affinity DataIC50: 38nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM476219(US10865384, Compound D4476 | US11633415, Compound ...)
Affinity DataIC50: 214nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717684(US12215095, Compound ZH3-90)
Affinity DataIC50: 269nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent

TargetCasein kinase I isoform delta(Human)
University of Melbourne

US Patent
LigandPNGBDBM717680(US12215095, Compound ZH2-66)
Affinity DataIC50: 1.38E+3nMAssay Description:The assay used was the HotSpot assay (Reaction Biology Corp).Compounds were tested in 10-dose IC50 mode with a 3-fold serial dilution starting at 10 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/10/2025
Entry Details
Go to US Patent