Compile Data Set for Download or QSAR
Report error Found 417 Enz. Inhib. hit(s) with all data for entry = 12625
LigandPNGBDBM716029((1R,3S)-4'-Chloro-5'-(3-(4-(cyanomethyl)-3- methyl...)
Affinity DataKi:  0.390nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715884((1R,3S)-5'-(4-Amino-3-(dimethylcarbamoyl)-2- fluor...)
Affinity DataKi:  0.810nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715985((R)-(6-Amino-3-(4'-chloro-1',2'- dihydrospiro[cycl...)
Affinity DataKi:  0.890nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716037((1R,3S)-5'-(3-Amino-5-(4-(cyanomethyl)-3- methylpy...)
Affinity DataKi:  0.900nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715912((1R,3S)-4'-Chloro-3-methyl-5'-(3-(1-methyl-2- oxo-...)
Affinity DataKi:  0.910nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715927(6-Amino-3-((1R,2R)-4'-chloro-2-isopropyl-1',2'- di...)
Affinity DataKi:  1.41nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715969(6-Amino-3-((1R,2S)-4'-chloro-2-methyl-1',2'- dihyd...)
Affinity DataKi:  1.73nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715814((1S,3R)-5'-(4-Amino-3-(dimethylcarbamoyl)-2- fluor...)
Affinity DataKi:  1.74nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715793((1R,3S)-5'-(4-amino-3-(dimethylcarbamoyl)-2- fluor...)
Affinity DataKi:  2.07nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715853(5'-(4-Amino-3-(dimethylcarbamoyl)-2- fluorophenyl)...)
Affinity DataKi:  2.08nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM50583346(CHEMBL5078234 | US12208088, Compound 37)
Affinity DataKi:  2.20nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715876(6-Amino-3-(4'-chloro-4-(4-methyl-1H-pyrazol-1- yl)...)
Affinity DataKi:  2.21nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715879(6-Amino-3-((1R,2R)-4'-chloro-2-ethyl-1',2'- dihydr...)
Affinity DataKi:  2.51nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715886(6-Amino-3-((1R,3S)-4'-chloro-3-methyl-3-(3- methyl...)
Affinity DataKi:  2.63nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715831(6-Amino-3-((1R,3S)-4'-chloro-3-(4-methyl-2H-1,2,3-...)
Affinity DataKi:  2.84nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715857(6-Amino-3-(3-(2-amino-2-oxoethyl)-4'-chloro- 1',2'...)
Affinity DataKi:  2.95nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716018(6-Amino-3-((1R,3R)-4'-chloro-3-(hydroxymethyl)- 1'...)
Affinity DataKi:  3nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716006(2-(2-(3-(1',2'-Dihydrospiro[cyclopropane-1,3'- pyr...)
Affinity DataKi:  3.15nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715797(6-Amino-2-fluoro-N,N-dimethyl-3-((1R,2R)2-methyl-1...)
Affinity DataKi:  3.25nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715878(6-Amino-3-((1R,2S)-4'-chloro-2-ethyl-1',2'- dihydr...)
Affinity DataKi:  3.30nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715845(6-Amino-3-(4'-chloro-3-(4-methyl-1H-pyrazol-1- yl)...)
Affinity DataKi:  3.56nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715938(6-Amino-3-((1R,2R)-4'-chloro-2-phenyl-1',2'- dihyd...)
Affinity DataKi:  3.58nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715926(6-Amino-3-((1R,2R)-4'-chloro-2-isopropyl-1',2'- di...)
Affinity DataKi:  3.64nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715933(6-Amino-3-((1R,2S)-4'-chloro-2-propyl-1',2'- dihyd...)
Affinity DataKi:  3.64nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715987((R)-(3-(4'-Chloro-1',2'-dihydrospiro[cyclopentane-...)
Affinity DataKi:  3.87nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716027((1R,3S)-4'-Chloro-5'-(3-(4-(cyanomethyl)-3- methyl...)
Affinity DataKi:  3.90nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715976(6-Amino-2-fluoro-3-((1R,2R)-2-isopropyl-1',2'- dih...)
Affinity DataKi:  3.92nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715852(6-Amino-3-(4'-chloro-3-cyano-3-methyl-1',2'- dihyd...)
Affinity DataKi:  3.93nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715851(6-Amino-3-(4'-chloro-3-(cyanomethyl)-1',2'- dihydr...)
Affinity DataKi:  4nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715906((R)-(3-(1',2'-dihydrospiro[cyclopropane-1,3'- pyrr...)
Affinity DataKi:  4.20nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716020(6-Amino-3-((1R,3S)-4'-chloro-3-cyano-3-methyl- 1',...)
Affinity DataKi:  4.20nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716003(2-(2-(3-(4'-Chloro-1',2'- dihydrospiro[cyclopentan...)
Affinity DataKi:  4.30nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715881(6-Amino-3-((1R,3S)-4'-chloro-3-cyano-3-ethyl- 1',2...)
Affinity DataKi:  4.35nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715896(6-Amino-3-(4'-chloro-1',2'- dihydrospiro[cycloprop...)
Affinity DataKi:  4.39nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715743(6-Amino-3-(4'-chloro-1',2'- dihydrospiro[cyclobuta...)
Affinity DataKi:  4.40nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715825(6-Amino-3-(3-(2-amino-2-oxoethylidene)-4'- chloro-...)
Affinity DataKi:  4.5nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715730(6-Amino-3-(4'-chloro-1',2'- dihydrospiro[cycloprop...)
Affinity DataKi:  4.70nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715937(6-Amino-3-(4'-chloro-1',2'- dihydrospiro[cyclohexa...)
Affinity DataKi:  4.76nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715968(6-Amino-3-((1R,2S)-4'-chloro-2-methyl-1',2'- dihyd...)
Affinity DataKi:  4.76nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716002(6-Amino-3-(4'-chloro-4-(hydroxymethyl)-1',2'- dihy...)
Affinity DataKi:  4.89nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715932(6-Amino-3-((1R,2S)-4'-chloro-2-propyl-1',2'- dihyd...)
Affinity DataKi:  5.13nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716009((6-Amino-3-((1s,4s)-4'-chloro-4-hydroxy-1',2'- dih...)
Affinity DataKi:  5.20nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715771(3-(3-(1S,3R)-4'-chloro-3-hydroxy-1',2'- dihydrospi...)
Affinity DataKi:  5.40nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715804(6-Amino-3-((1R,3S)-4'-chloro-3-cyano-1',2'- dihydr...)
Affinity DataKi:  5.53nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715900(6-Amino-3-((1R,3S)-4'-chloro-3-(4-ethyl-1H- pyrazo...)
Affinity DataKi:  5.54nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715992(6-Amino-3-((1R,2S)-2-ethyl-1',2'- dihydrospiro[cyc...)
Affinity DataKi:  5.78nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716007(2-(2-(3-(4'-Chloro-1',2'- dihydrospiro[cyclopentan...)
Affinity DataKi:  5.94nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM715800(6-Amino-3-((1R,3S)-4'-chloro-3-(2H-1,2,3-triazol-2...)
Affinity DataKi:  6nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716001(6-Amino-3-(4'-chloro-4-(hydroxymethyl)-1',2'- dihy...)
Affinity DataKi:  6.01nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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LigandPNGBDBM716017(6-Amino-3-((1R,3S)-4'-chloro-3-(hydroxymethyl)- 1'...)
Affinity DataKi:  6.10nMAssay Description:For the binding assay, 4 ul 2×HPK1 and Eu-anti-GST antibody were added to each well of the assay plate using a Multidrop reagent dispenser. The solut...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
6/3/2025
Entry Details
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