Compile Data Set for Download or QSAR
Report error Found 29 Enz. Inhib. hit(s) with all data for entry = 12609
TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713684(2,4,6-trimethyl-N-[2-(2- methylphenyl)ethyl]benzen...)
Affinity DataIC50: 90nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713680(N-[2-(2-chlorophenyl)ethyl]-2,4,6- trimethylbenzen...)
Affinity DataIC50: 270nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713681(N-[2-(2-bromophenyl)ethyl]-2,4,6- trimethylbenzene...)
Affinity DataIC50: 270nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713685(4-bromo-2,6-dichloro-N-[2-(2- methylphenyl)ethyl]b...)
Affinity DataIC50: 270nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713696(N-[2-(2-chlorophenyl)ethyl]-4-methoxy-2,6- dimethy...)
Affinity DataIC50: 300nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713694(4-bromo-2,6-dichloro-N-[2-(2- hydroxyphenyl)ethyl]...)
Affinity DataIC50: 300nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713688(2,6-dichloro-N-[2-(2-chlorophenyl)ethyl]-4- cyclop...)
Affinity DataIC50: 360nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 1(Human)
Glucox Biotech

US Patent
LigandPNGBDBM50330722(2-(2-chlorophenyl)-4-methyl-5-(pyridin-2-ylmethyl)...)
Affinity DataIC50: 500nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713693(N-[2-(2-hydroxyphenyl)ethyl]-2,4,6- trimethylbenze...)
Affinity DataIC50: 800nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713698(4-hydroxy-N-[2-(2-hydroxyphenyl)ethyl]- 2,6-dimeth...)
Affinity DataIC50: 870nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713693(N-[2-(2-hydroxyphenyl)ethyl]-2,4,6- trimethylbenze...)
Affinity DataIC50: 900nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713686(4-bromo-2,6-dichloro-N-[2-(2- chlorophenyl)ethyl]b...)
Affinity DataIC50: 900nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713695(6-chloro-3-hydroxy-N-[2-(2- hydroxyphenyl)ethyl]-2...)
Affinity DataIC50: 900nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713697(N-[2-(2-hydroxyphenyl)ethyl]-4-methoxy- 2,6-dimeth...)
Affinity DataIC50: 1.00E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713687(2,6-dichloro-4-cyclopropyl-N-[2-(2- fluorophenyl)e...)
Affinity DataIC50: 1.10E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713694(4-bromo-2,6-dichloro-N-[2-(2- hydroxyphenyl)ethyl]...)
Affinity DataIC50: 1.50E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713689(2,6-dichloro-N-[2-(2-chlorophenyl)ethyl]-4- (trifl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713682(N-[2-(2-chlorophenyl)ethyl]-2,2,4,6,7- pentamethyl...)
Affinity DataIC50: 1.60E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM50330722(2-(2-chlorophenyl)-4-methyl-5-(pyridin-2-ylmethyl)...)
Affinity DataIC50: 1.60E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713697(N-[2-(2-hydroxyphenyl)ethyl]-4-methoxy- 2,6-dimeth...)
Affinity DataIC50: 1.60E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713691(US12202790, Example 35 isomer 1)
Affinity DataIC50: 1.70E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713690(4-bromo-2,6-dichloro-N-[2-fluoro-2-(2- methylpheny...)
Affinity DataIC50: 1.70E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713679(N-[2-(2-fluorophenyl)ethyl]-2,4,6- trimethylbenzen...)
Affinity DataIC50: 2.20E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713683(2-chloro-6-methyl-N-[2-(2- methylphenyl)ethyl]benz...)
Affinity DataIC50: 2.40E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713695(6-chloro-3-hydroxy-N-[2-(2- hydroxyphenyl)ethyl]-2...)
Affinity DataIC50: 2.40E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713692(US12202790, Example 35 isomer 2)
Affinity DataIC50: 4.90E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetCytochrome b-245 heavy chain(Human)
Glucox Biotech

US Patent
LigandPNGBDBM50330722(2-(2-chlorophenyl)-4-methyl-5-(pyridin-2-ylmethyl)...)
Affinity DataIC50: 9.00E+3nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 4(Human)
Glucox Biotech

US Patent
LigandPNGBDBM713698(4-hydroxy-N-[2-(2-hydroxyphenyl)ethyl]- 2,6-dimeth...)
Affinity DataIC50: 2.20E+4nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent

TargetNADPH oxidase 5(Human)
Glucox Biotech

US Patent
LigandPNGBDBM50330722(2-(2-chlorophenyl)-4-methyl-5-(pyridin-2-ylmethyl)...)
Affinity DataIC50: 4.40E+4nMAssay Description:Reactive oxygen produced in whole cells or in membrane preparation of Nox1, Nox3, Nox4, Nox5 and xanthine oxidase and glucose oxidase were determined...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/29/2025
Entry Details
Go to US Patent