Compile Data Set for Download or QSAR
Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 12495
TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706739(US12157739, Example 1)
Affinity DataIC50: 90nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706745(US12157739, Example 29)
Affinity DataIC50: 370nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706747(US12157739, Example 75)
Affinity DataIC50: 420nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706743(US12157739, Example 11)
Affinity DataIC50: 440nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706742(US12157739, Example 4)
Affinity DataIC50: 530nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706746(US12157739, Example 35)
Affinity DataIC50: 590nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706744(US12157739, Example 12)
Affinity DataIC50: 610nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706740(US12157739, Example 2)
Affinity DataIC50: 640nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
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TargetEgl nine homolog 1 [184-418](Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM706741(US12157739, Example 3)
Affinity DataIC50: 640nMAssay Description:An enzyme (human PHD2 184-418) and the substrate were diluted with an assay buffer (pH 7.4) containing 10 mM HEPES, 150 mM NaCl, 10 μM MnCl2-4H2O, 2 ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
4/14/2025
Entry Details
Go to US Patent