Compile Data Set for Download or QSAR
Report error Found 60 Enz. Inhib. hit(s) with all data for entry = 12173
TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684577(US12030897, Example 32)
Affinity DataIC50: 2nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684574(US12030897, Example 25)
Affinity DataIC50: 2nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 2nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684576(US12030897, Example 31)
Affinity DataIC50: 3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 4nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684568(US12030897, Example 18)
Affinity DataIC50: 4nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 6nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684569(US12030897, Example 20)
Affinity DataIC50: 7nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684567(US12030897, Example 16)
Affinity DataIC50: 7nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684564(US12030897, Example 7)
Affinity DataIC50: 10nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684565(US12030897, Example 8)
Affinity DataIC50: 10nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684566(US12030897, Example 9)
Affinity DataIC50: 11nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684560(US12030897, Example 4)
Affinity DataIC50: 12nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684575(US12030897, Example 30)
Affinity DataIC50: 14nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684562(US12030897, Example 5)
Affinity DataIC50: 16nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684563(US12030897, Example 6)
Affinity DataIC50: 18nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-2(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684561(US12030897, Example 1)
Affinity DataIC50: 24nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 41nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 61nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 109nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 139nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684563(US12030897, Example 6)
Affinity DataIC50: 150nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684560(US12030897, Example 4)
Affinity DataIC50: 156nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684560(US12030897, Example 4)
Affinity DataIC50: 161nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684569(US12030897, Example 20)
Affinity DataIC50: 167nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684565(US12030897, Example 8)
Affinity DataIC50: 184nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684566(US12030897, Example 9)
Affinity DataIC50: 201nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684574(US12030897, Example 25)
Affinity DataIC50: 207nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684569(US12030897, Example 20)
Affinity DataIC50: 230nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684577(US12030897, Example 32)
Affinity DataIC50: 284nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 306nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684566(US12030897, Example 9)
Affinity DataIC50: 325nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684577(US12030897, Example 32)
Affinity DataIC50: 356nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684574(US12030897, Example 25)
Affinity DataIC50: 369nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684565(US12030897, Example 8)
Affinity DataIC50: 385nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 438nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684568(US12030897, Example 18)
Affinity DataIC50: 509nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684567(US12030897, Example 16)
Affinity DataIC50: 535nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684575(US12030897, Example 30)
Affinity DataIC50: 663nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684576(US12030897, Example 31)
Affinity DataIC50: 667nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684563(US12030897, Example 6)
Affinity DataIC50: 743nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684567(US12030897, Example 16)
Affinity DataIC50: 861nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 909nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684561(US12030897, Example 1)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684576(US12030897, Example 31)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684575(US12030897, Example 30)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684561(US12030897, Example 1)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetReceptor tyrosine-protein kinase erbB-4(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684570(US12030897, Example 21 | US12030897, Example 23 | ...)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

TargetEpidermal growth factor receptor(Human)
Medshine Discovery

US Patent
LigandPNGBDBM684562(US12030897, Example 5)
Affinity DataIC50: 1.00E+3nMAssay Description:The object of this test is to detect the in vitro inhibitory activity of the compound against HER1 (ErbB1), HER2 (ErbB2) and HER4 (ErbB4). The enzyme...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2024
Entry Details
Go to US Patent

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