Compile Data Set for Download or QSAR
Report error Found 13 Enz. Inhib. hit(s) with all data for entry = 11715
TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM642525(US11851436, Compound A1-8)
Affinity DataIC50: 15.7nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM642526(US11851436, Compound A1-9)
Affinity DataIC50: 17.8nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568105(CHEMBL4858455 | US11851436, Compound A1-3)
Affinity DataIC50: 18.4nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM25017(2-[(3,5-difluoro-4-hydroxyphenyl)amino]-5,7-dimeth...)
Affinity DataIC50: 22.6nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568104(CHEMBL4858257 | US11851436, Compound A1-2)
Affinity DataIC50: 24.6nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568110(CHEMBL4865383 | US11851436, Compound A1-11)
Affinity DataIC50: 25.7nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568111(CHEMBL4878141 | US11851436, Compound A1-12)
Affinity DataIC50: 34.7nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM642518(US11851436, Compound A1-1)
Affinity DataIC50: 55.5nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568107(CHEMBL4845736 | US11851436, Compound A1-6)
Affinity DataIC50: 79.8nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568108(CHEMBL4860957 | US11851436, Compound A1-7)
Affinity DataIC50: 81.8nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568109(CHEMBL4861235 | US11851436, Compound A1-10)
Affinity DataIC50: 95.8nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM642522(US11851436, Compound A1-5)
Affinity DataIC50: 148nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
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TargetRibosomal protein S6 kinase alpha-3(Human)
University of Colorado

US Patent
LigandPNGBDBM50568106(CHEMBL4849660 | US11851436, Compound A1-4)
Affinity DataIC50: 329nMAssay Description:LANCE (Lanthanide Chelate Excite) Eu time-resolved fluorescence resonance energy transfer (TR-FRET) kinase assay (PerkinElmer) was performed in 384-w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/15/2024
Entry Details
Go to US Patent