Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 11708
TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642197BDBM642197(US1184575, 14-acetyl oxycodone)
Affinity DataKi:  18nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642198BDBM642198(US1184575, 6-PEG oxycodone)
Affinity DataKi:  22nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 50370595BDBM50370595(US9233167, Oxycodone | Oxycontin | OXYCODONE | US1...)
Affinity DataKi:  30nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642196BDBM642196(US1184575, 6-acetyl oxycodone)
Affinity DataKi:  41nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642199BDBM642199(US1184575, 6,14-bis-PEG oxycodone)
Affinity DataKi:  52nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642200BDBM642200(US1184575, 6-lauroyl oxycodone)
Affinity DataKi:  96nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642201BDBM642201(US1184575, 14-lauroyl oxycodone)
Affinity DataKi:  160nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent

TargetMu-type opioid receptor(Human)
Rhodes Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 642202BDBM642202(US1184575, 6,14-bis-lauroyl oxycodone)
Affinity DataKi:  2.22E+4nMAssay Description:Radioligand dose-displacement binding assays for μ-opioid receptors can use 0.3 nM [3H]-diprenorphine (Perkin Elmer, Shelton, CT), with 5 mg mem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2024
Entry Details
US Patent