Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 11571
TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 75.1nMAssay Description:Table 9: Human LOX amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
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TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 209nMAssay Description:Table 9: The amine oxidase activity was evaluated by measuring Amplex Red fluorescence using commercially available purified, recombinant human LOXL2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461420(US11072585, Example 12 | BDBM509178 | US10774069, ...)
Affinity DataIC50: 300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461386(US10774069, Compound Rac-1 | US11072585, Example 1...)
Affinity DataIC50: 300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetLysyl oxidase homolog 2(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 300nMAssay Description:Table 8: LOXL2 amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (non BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetLysyl oxidase homolog 3(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 1.21E+3nMAssay Description:Table 9: The amine oxidase activity was evaluated by measuring Amplex Red fluorescence using commercially available purified, recombinant human LOXL3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent

TargetProtein-lysine 6-oxidase (LOX)(Human)
Pharmakea

US Patent
LigandPNGBDBM461421(US10774069, Compound 1 | US11072585, Example 120 |...)
Affinity DataIC50: 4.70E+4nMAssay Description:Table 9: Human LOX amine oxidase activity was evaluated by measuring Amplex Red fluorescence using 10-20× concentrated conditioned media (BSA-contain...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2023
Entry Details
Go to US Patent