Compile Data Set for Download or QSAR
Report error Found 317 Enz. Inhib. hit(s) with all data for entry = 11190
TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598223(US11612606, Compound 555b | (3R,4S)-4-Methyltetrah...)
Affinity DataIC50: 24nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598131(US11612606, Compound 484b | (1r,3r)-3-Cyanocyclobu...)
Affinity DataIC50: 26nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598255(US11612606, Compound 574a | (1r,3r)-3-(2-Hydroxypr...)
Affinity DataIC50: 32nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598083(US11612606, Compound 441b | amino-7-fluoro-6-(8-me...)
Affinity DataIC50: 36nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598127(US11612606, Compound 482a | (trans)-2-Cyanocyclope...)
Affinity DataIC50: 38nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598330(US11612606, Compound 751 | N-(8-Amino-7-fluoro-6-(...)
Affinity DataIC50: 41nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598334(US11612606, Compound 755 | N-(8-Amino-7-fluoro-6-(...)
Affinity DataIC50: 46nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598031(US11612606, Compound 403a | (R)-Tetrahydrofuran-3-...)
Affinity DataIC50: 48nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
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TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598148(US11612606, Compound 510c | 1H-pyrido[2,3-b][1,4]o...)
Affinity DataIC50: 62nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598210(US11612606, Compound 546a | trans-4-Methoxytetrahy...)
Affinity DataIC50: 62nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598336(US11612606, Compound 527 | 3-Hydroxy-3-methylcyclo...)
Affinity DataIC50: 64nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598117(US11612606, Compound 477d | amino-7-fluoro-6-(8-me...)
Affinity DataIC50: 66nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

TargetLymphocyte cytosolic protein 2(Human)
Genentech

US Patent
LigandPNGBDBM598027(US11612606, Compound 401 | Tetrahydro-2H-pyran-4-y...)
Affinity DataIC50: 97nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598031(US11612606, Compound 403a | (R)-Tetrahydrofuran-3-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598056(US11612606, Compound 417 | 2-Methyl-2-azaspiro[3.3...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598057(US11612606, Compound 418a | (R)-1-Acetylpyrrolidin...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598059(US11612606, Compound 420 | 1-(2,2,2-Trifluoroethyl...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598060(US11612606, Compound 421 | 1-(Oxetan-3-yl)piperidi...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598062(US11612606, Compound 423 | 7-Methyl-7-azaspiro[3.5...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598063(US11612606, Compound 424 | 2-Acetyl-2-azaspiro[3.3...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598064(US11612606, Compound 425 | 2-Methyl-2-azaspiro[3.3...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598065(US11612606, Compound 426 | 1-Acetylazetidin-3-yl(8...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598066(US11612606, Compound 427 | 7-Methyl-7-azaspiro[3.5...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598067(US11612606, Compound 428 | 6-Methyl-6-azaspiro[3.4...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598069(US11612606, Compound 430 | 7-(Oxetan-3-yl)-7-azasp...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598071(US11612606, Compound 432a | (1R,5S,6r)-3-Methyl-3-)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598072(US11612606, Compound 433 | (cis)-3-Fluoro-1-methyl...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598073(US11612606, Compound 434 | 1-(2,2-Difluoroethypaze...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598076(US11612606, Compound 437a | (3S,4R)-1-Acetyl-3-flu...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598078(US11612606, Compound 439a | (1R,5S,9s)-7-Methyl-3-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598082(US11612606, Compound 441a | (trans)-4-Methyltetrah...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598083(US11612606, Compound 441b | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598090(US11612606, Compound 443 | 2-(Oxetan-3-yl)-2-azasp...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598091(US11612606, Compound 444a | (S)-1-Methyl-5-oxopyrr...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598092(US11612606, Compound 444b | amino-6-(8-ethyl-2,3-d...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598093(US11612606, Compound 445ab | (+1-)-trans-3-Fluoro-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598095(US11612606, Compound 445d | yl(8-amino-7-fluoro-6-...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598096(US11612606, Compound 447a | (1r,3r)-3-(Dimethylami...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598099(US11612606, Compound 451b | yl)methyl(8-amino-7-fl...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598103(US11612606, Compound 452d | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598111(US11612606, Compound 467d | azaspiro[4.4]nonan-3-y...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598119(US11612606, Compound 478b | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598122(US11612606, Compound 479b | amino-7-fluoro-6-(8-me...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598127(US11612606, Compound 482a | (trans)-2-Cyanocyclope...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598128(US11612606, Compound 482b | fluoro-6-(8-methyl-2,3...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598129(US11612606, Compound 483a | (1s,3s)-3-cyanocyclobu...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598130(US11612606, Compound 484a | (1s,3s)-3-Cyanocyclobu...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598132(US11612606, Compound 485a | (1s,3s)-3-Hydroxycyclo...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598133(US11612606, Compound 485b | (1r,3r)-3-Hydroxycyclo...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

LigandPNGBDBM598134(US11612606, Compound 486 | 3-Hydroxy-3-methylcyclo...)
Affinity DataKi: <0.0130nMAssay Description:TBDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/9/2023
Entry Details
Go to US Patent

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