Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 11159
TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552714(CHEMBL4749593 | US11591329, Ex. No. 2)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595677(US11591329, Ex. No. 4 | 3-Methyl-8-(3-(1-methyl-1H...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552715(CHEMBL4753114 | US11591329, Ex. No. 5)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595679(US11591329, Ex. No. 6 | 3-Ethyl-1-methyl-4-(3-(1-m...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552719(CHEMBL4780804 | US11591329, Ex. No. 19)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595691(US11591329, Ex. No. 18 | 4-(3-(3-Fluoro-4-(4-methy...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552718(CHEMBL4740345 | US11591329, Ex. No. 16)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552717(CHEMBL4798507 | US11591329, Ex. No. 15)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595685(US11591329, Ex. No. 12 | 1-Methyl-4-(3-(1-methyl-1...)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM50552716(CHEMBL4754734 | US11591329, Ex. No. 13)
Affinity DataIC50: 10nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595687(US11591329, Ex. No. 14 | 1-Cyclopropyl-3-methyl-4-...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595694(US11591329, Ex. No. 21 | 4-(6-Chloro-3-(1-methyl-1...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595690(US11591329, Ex. No. 17 | 3-Isopropyl-1-methyl-4-(3...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595682(US11591329, Ex. No. 9 | 3-(Cyclopropylmethyl)-1-me...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595681(US11591329, Ex. No. 8 | 3-Benzyl-1-methyl-4-(3-(1-...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595680(US11591329, Ex. No. 7 | 3,3-Diethyl-1-methyl-4-(3-...)
Affinity DataIC50: 20nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595693(US11591329, Ex. No. 20 | 3-Isopropyl-1-methyl-4-(3...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595695(US11591329, Ex. No. 22 | 1,3-Dimethyl-4-(6-methyl-...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595696(US11591329, Ex. No. 23 | 5-(2,4-Dimethyl-3-oxopipe...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595697(US11591329, Ex. No. 24 | 4-(6-Methoxy-3-(1-methyl-...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595698(US11591329, Ex. No. 25 | 4-(6-(Furan-3-yl)-3-(1-me...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595699(US11591329, Ex. No. 26 | 4-(6-Benzyl-3-(1-methyl-1...)
Affinity DataIC50: 115nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595674(US11591329, Ex. No. 1 | 1-(3-(1-Methyl-1H-pyrazol-...)
Affinity DataIC50: 200nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
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Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595684(US11591329, Ex. No. 11 | 1-Methyl-4-(3-(1-methyl-1...)
Affinity DataIC50: 200nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595683(US11591329, Ex. No. 10 | 1-Methyl-4-(3-(1-methyl-1...)
Affinity DataIC50: 200nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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TargetFibroblast growth factor receptor 3(Human)
Incyte

US Patent
LigandPNGBDBM595676(US11591329, Ex. No. 3 | 5-(6,7-Dihydropyrazolo[1,5...)
Affinity DataIC50: 200nMAssay Description:The inhibitor potency of the exemplified compounds was measured in an enzyme assay that measures peptide phosphorylation using FRET measurements to d...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/14/2023
Entry Details
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