Compile Data Set for Download or QSAR
Report error Found 195 Enz. Inhib. hit(s) with all data for entry = 11059
LigandPNGBDBM588211(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
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Date in BDB:
2/26/2023
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LigandPNGBDBM588211(methyl 4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cycl...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
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Date in BDB:
2/26/2023
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LigandPNGBDBM588212(4-[4-[[1-[(4- fluorophenyl)carbamoyl]- cyclopropan...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588213(1-N-[4-(6-carbamoyl-7- methoxyquinolin-4- yl)oxyph...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
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Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
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Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588214(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- (methy...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoPurchaseSimilars
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Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588215(1-N-[4-[6-[2- (dimethylamino)ethylcarbamoyl]- 7-me...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588215(1-N-[4-[6-[2- (dimethylamino)ethylcarbamoyl]- 7-me...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
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LigandPNGBDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588216(1-N'-(4-fluorophenyl)-N-[4-[7- methoxy-6-(2-piperi...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588217(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(2-morp...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588218(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(oxetan...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
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In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588218(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(oxetan...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588219(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [(1-me...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588219(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [(1-me...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588220(1-N-[4-[6-(azetidine-1- carbonyl)-7-methoxyquinoli...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588221(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588221(1-N'-(4-fluorophenyl)-1-N- [4-[6-(3-hydroxyazetidi...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588222(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2R)...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588223(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6- [[(2S)...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588224(1-N-[4-(6-cyano-7- methoxyquinolin-4- yl)oxyphenyl...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588225(1-N'-(4-fluorophenyl)-1-N- [4-[7-methoxy-6-(1,3-ox...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588232(1-N-[4-[6-carbamoyl-7-(3- morpholin-4- ylpropoxy)q...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588233(1-N-[4-[6-carbamoyl-7-(2- methoxyethoxy)quinolin-4...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588233(1-N-[4-[6-carbamoyl-7-(2- methoxyethoxy)quinolin-4...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588234(methyl 4-[2-chloro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588234(methyl 4-[2-chloro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588234(methyl 4-[2-chloro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588236(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588236(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588236(1-N'-[4-(6-carbamoyl-7- methoxyquinolin-4-yl)oxy-3...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588237(1-N'-[3-chloro-4-[7-methoxy-6 (methylcarbamoyl)qui...)
Affinity DataIC50: 10nMAssay Description:Human Met (residues R974-S1390 with A1209G and V1290L, 3.4 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKKGQEEEYVFIE (SEO ID NO...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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LigandPNGBDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Axl (residues H473-A894 with Q764R, 161 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 250 μM KKSRGDYMTMQIG (SEO ID NO. 43) 10 mM m...More data for this Ligand-Target Pair
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Date in BDB:
2/26/2023
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LigandPNGBDBM588238(methyl 4-[2-fluoro-4-[[1-[(4- fluorophenyl)carbamo...)
Affinity DataIC50: 10nMAssay Description:Human Mer (residues R557-E882 with H628Q and R794A, 0.7 nM) was incubated with 8 mM MOPS pH 7.0, 0.2 mM EDTA, 30 mM NaCl, 250 μM GGMEDIYFEFMGGKK...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
2/26/2023
Entry Details
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